SCHEMBL9434600

SCHEMBL9434600

CC(O)(c1cccc(O)c1)c1nccs1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.44
ALOX5 P09917 14/20 0.41
PRKDC P78527 1/20 0.37
CASR P41180 1/20 0.36
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813254 0.81 ALOX5 (0.60) ALOX5
SCHEMBL9369962 0.81 ALOX5 (0.60) ALOX5
SCHEMBL9434229 0.79 AR (0.55) KCNH2ALOX5PRKDC
SCHEMBL9433089 0.77 ALOX5 (0.45) KCNH2ALOX5PRKDCCASR
SCHEMBL8682794 0.76 ALDH1A1 (0.40) KCNH2ALOX5PRKDC
SCHEMBL8614144 0.76 KCNH2 (0.38) KCNH2ALOX5PRKDCCASR
SCHEMBL29605276 0.75 KCNH2 (0.41) KCNH2ALOX5PRKDC
SCHEMBL31584832 0.74 CASR (0.46) KCNH2ALOX5PRKDCCASR
SCHEMBL8612881 0.73 AR (0.36) KCNH2ALOX5PRKDC
SCHEMBL2984624 0.73 KCNH2 (0.41) KCNH2ALOX5PRKDCCASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283245-A Antiinflammatory agent, antiallergens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-02-01 US disclosed
US-5089495-A Lipoxygenase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (FR) 1992-02-18 US disclosed
EP-0381375-A1 Heterocyclic derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-08-08 EP disclosed