SCHEMBL9436730

SCHEMBL9436730

COC(=S)c1ccc(-c2ccccc2)c(S(C)(=O)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.50
ROCK2 O75116 1/20 0.45
TDP1 Q9NUW8 1/20 0.43
EGFR P00533 1/20 0.43
LOXL2 Q9Y4K0 2/20 0.41
ACLY P53396 2/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
ITGAV P06756 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796477 0.80 TDP1 (0.50) PTGS2ROCK2TDP1LOXL2ACLY
SCHEMBL9167776 0.79 EGFR (0.56) PTGS2EGFR
SCHEMBL9189128 0.78 SLC9A1 (0.46) LOXL2
SCHEMBL16618470 0.78 PTGS2 (0.47) PTGS2ROCK2LOXL2ACLY
SCHEMBL9189120 0.78 PTGS2 (0.40) PTGS2ROCK2TDP1LOXL2ACLY
SCHEMBL11665324 0.77 EGFR (0.44) PTGS2EGFR
SCHEMBL9166737 0.77 ESR2 (0.51) PTGS2ROCK2EGFR
Hydrochloric Acid SCHEMBL9436715 0.77 SLC9A1 (0.45) LOXL2
SCHEMBL8895570 0.77 PTGS2 (0.60) PTGS2ROCK2EGFRACLY
Hydrochloric Acid SCHEMBL9192121 0.77 LOXL2 (0.41) PTGS2ROCK2TDP1LOXL2ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292755-A USPA benzolyguanidines HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-08 US disclosed
US-5091394-A BENZOYLGUANIDINES, A PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-25 US disclosed