SCHEMBL9437726

SCHEMBL9437726

CN(CCN)CCCCc1ccc2c(c1)OCC(=O)N2C

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.51
HTR2C P28335 3/20 0.48
SMPD1 P17405 1/20 0.42
NMT1 P30419 3/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
SLC6A4 P31645 1/20 0.42
KCNH2 Q12809 1/20 0.42
GABRA1 P14867 1/20 0.41
GABRA5 P31644 1/20 0.41
CYP11B2 P19099 2/20 0.40
CYP11B1 P15538 1/20 0.40
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
PRKCQ Q04759 1/20 0.37
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437707 0.87 HTR1A (0.57) HTR1AHTR2CNMT1HTR1DHTR1B
SCHEMBL9437818 0.85 HTR1A (0.49) HTR1AHTR2CSMPD1NMT1HTR1D
SCHEMBL9437796 0.85 HTR1A (0.54) HTR1AHTR2CHTR1DHTR1BSLC6A4
SCHEMBL9437724 0.83 HTR1A (0.55) HTR1AHTR2CNMT1HTR1DHTR1B
SCHEMBL9437846 0.80 HTR1A (0.46) HTR1AHTR2CNMT1HTR1DHTR1B
SCHEMBL8786888 0.80 HTR1A (0.57) HTR1AHTR2CNMT1HTR1DHTR1B
SCHEMBL9437864 0.79 HTR1A (0.43) HTR1AHTR2CSMPD1NMT1HTR1D
SCHEMBL9437737 0.78 HTR1A (0.55) HTR1AHTR2CNMT1HTR1DHTR1B
SCHEMBL8177698 0.76 HTR1A (0.48) HTR1AHTR2CSMPD1NMT1HTR1D
SCHEMBL8785675 0.76 HTR1A (0.55) HTR1AHTR2CNMT1HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed