SCHEMBL9437792

SCHEMBL9437792

NCCc1ccc2c(c1)OCC(=O)N2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 9/20 0.53
DRD3 P35462 9/20 0.53
DRD2 P14416 8/20 0.53
PARP1 P09874 3/20 0.52
HTR1A P08908 2/20 0.51
NR3C2 P08235 2/20 0.51
CHRM5 P08912 1/20 0.51
ADRA2A P08913 1/20 0.51
ADRA2B P18089 1/20 0.51
HTR2A P28223 1/20 0.51
ADRA1B P35368 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
TAAR1 Q96RJ0 1/20 0.49
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
MMP12 P39900 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437898 0.88 PARP1 (0.68) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL8191537 0.88 DRD4 (0.55) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL8195715 0.85 PARP1 (0.60) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL9437789 0.85 DRD4 (0.53) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL3777130 0.81 DRD4 (0.55) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL2056366 0.81 PARP1 (0.77) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL6329957 0.81 DRD4 (0.53) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL276741 0.79 MMP12 (0.51) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL29512901 0.79 MMP12 (0.51) DRD4DRD3DRD2PARP1HTR1A
SCHEMBL27590225 0.78 TP53 (0.47) DRD4DRD3DRD2PARP1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5225409-A Serotoninergic disorders; anxiolytic agents; schizophrenia ADIR ET COMPAGNIE (FR) 1993-07-06 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed