SCHEMBL9439381

SCHEMBL9439381

CCOC(=O)C[CH]Oc1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
ALDH1A1 P00352 5/20 0.48
HPGD P15428 3/20 0.48
CDC25B P30305 2/20 0.47
BTN3A1 O00481 1/20 0.46
KDM4E B2RXH2 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAPK1 P28482 2/20 0.44
HSD17B10 Q99714 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PGR P06401 1/20 0.44
GAA P10253 1/20 0.44
PTGS1 P23219 1/20 0.44
CDC25A P30304 1/20 0.44
CDC25C P30307 1/20 0.44
MITF O75030 1/20 0.44
LMNA P02545 1/20 0.44
HSP90AA1 P07900 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6707308 0.87 TNF (0.46) TSHRALDH1A1HPGDCDC25BBTN3A1
SCHEMBL7277411 0.83 ALDH1A1 (0.51) ALDH1A1HPGDKDM4ETDP1MAPK1
SCHEMBL7278827 0.83 ALDH1A1 (0.51) TSHRALDH1A1HPGDBTN3A1KDM4E
SCHEMBL11490448 0.79 TSHR (0.67) TSHRALDH1A1HPGDKDM4ETDP1
SCHEMBL31520212 0.79 TSHR (0.67) TSHRALDH1A1HPGDKDM4ETDP1
SCHEMBL15941488 0.78 TSHR (0.48) TSHRALDH1A1HPGDCDC25BKDM4E
SCHEMBL27493266 0.78 ALDH1A1 (0.53) TSHRALDH1A1HPGDCDC25BBTN3A1
SCHEMBL3861740 0.77 HTR1B (0.47) TSHRALDH1A1HPGDKDM4ETDP1
SCHEMBL9439384 0.77 KDM4E (0.56) TSHRALDH1A1HPGDKDM4ETDP1
SCHEMBL845701 0.75 KMT2A (0.62) ALDH1A1HPGDCDC25BKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278148-A Hypotensive agents HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
US-5250517-A Hypotensive and cardiotonic agents; cardiac insufficiency HOFFMANN-LA ROCHE INC. (US) 1993-10-05 US disclosed
US-5140011-A Hypotensive agents HOFFMANN-LA ROCHE, INC. (US) 1992-08-18 US disclosed
US-4931591-A Novel 5-amino-4-hydroxyvaleryl derivatives CIBA-GEIGY CORPORATION (US) 1990-06-05 US disclosed
US-4727060-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1988-02-23 US disclosed