SCHEMBL9439714

SCHEMBL9439714

Nc1nc(N)c2c(n1)NCC2CCCCCCC(=O)N[C@@H](CCC(=O)O)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GART P22102 9/20 0.46
ATIC P31939 5/20 0.45
TYMS P04818 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9439835 1.00 GART (0.46) GARTATICTYMS
SCHEMBL9439737 0.99 GART (0.45) GARTATICTYMS
SCHEMBL9439643 0.82 KMT2A (0.55)
SCHEMBL9439648 0.82 KMT2A (0.55)
SCHEMBL9439958 0.82 GART (0.38) GARTATIC
SCHEMBL8997257 0.81 GART (0.61) GARTATIC
SCHEMBL9439570 0.80 GART (0.58) GARTATIC
SCHEMBL9220611 0.80 MTHFD1 (0.56) GARTATIC
SCHEMBL9227822 0.79 DHFR (0.52) GARTATIC
SCHEMBL9227797 0.79 DHFR (0.57) GARTATICTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
EP-0418924-A2 Pyrrolopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-03-27 EP disclosed