SCHEMBL9439773

SCHEMBL9439773

COC(=O)c1ccc(C(C=O)=Cc2cn(Cc3ccccc3)c3nc(N)n(COC(C)C)c(=O)c23)s1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2L11 O43521 2/20 0.34
BCL2 P10415 2/20 0.34
BID P55957 2/20 0.34
BCL2L1 Q07817 2/20 0.34
MCL1 Q07820 2/20 0.34
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
APP P05067 1/20 0.33
SNCA P37840 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 2/20 0.33
CNR2 P34972 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
THRB P10828 1/20 0.31
P2RX7 Q99572 2/20 0.31
CFTR P13569 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9439775 0.81 KDM4E (0.33) SMN1; SMN2KDM4EKMT2ACA12CA1
SCHEMBL8997137 0.81 BRD4 (0.36) LMNASMN1; SMN2P2RX7
SCHEMBL8997174 0.79 PDE4A (0.38) ALDH1A1SMN1; SMN2KDM4EKMT2ACNR2
SCHEMBL9844748 0.74 DRD2 (0.39) ALDH1A1KDM4EKMT2ATHRBP2RX7
SCHEMBL9844781 0.66 DRD2 (0.40) ALDH1A1KDM4EKMT2ATHRBCFTR
SCHEMBL9844745 0.64 MAPT (0.35) ALDH1A1LMNASMN1; SMN2KDM4EKMT2A
SCHEMBL9439746 0.59 PTGER4 (0.34) HPGD
SCHEMBL10068017 0.57 CYP1A2 (0.50) ALDH1A1SMN1; SMN2KDM4EKMT2ACA12
SCHEMBL699995 0.54 APP (0.50) ALDH1A1LMNAAPPSNCASMN1; SMN2
SCHEMBL6030810 0.54 HDAC3 (0.76) ALDH1A1LMNAKDM4EPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed