SCHEMBL9844781

SCHEMBL9844781

COC(=O)c1ccc(CCc2c(Br)n(Cc3ccccc3)c3nc(N)n(COC(C)C)c(=O)c23)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.40
TBXA2R P21731 2/20 0.40
MAPK8 P45983 3/20 0.40
CFTR P13569 1/20 0.40
TLR7 Q9NYK1 3/20 0.38
MAPT P10636 3/20 0.38
THRB P10828 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
PKM P14618 1/20 0.37
TP53 P04637 1/20 0.36
OPRK1 P41145 1/20 0.36
GPR18 Q14330 1/20 0.36
P2RX3 P56373 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844748 0.85 DRD2 (0.39) DRD2TBXA2RCFTRTLR7MAPT
SCHEMBL9556787 0.80 DRD2 (0.45) DRD2TBXA2RMAPK8CFTRTLR7
SCHEMBL2072670 0.75 DRD2 (0.40) DRD2CFTRTLR7MAPTKDM4E
SCHEMBL1386593 0.75 DRD2 (0.40) DRD2CFTRTLR7MAPTKDM4E
SCHEMBL8997174 0.75 PDE4A (0.38) CFTRTLR7MAPTTHRBKDM4E
SCHEMBL9844802 0.70 AGTR1 (0.40) DRD2TBXA2RTLR7MAPTTHRB
SCHEMBL9844763 0.68 NPC1 (0.36) DRD2TLR7MAPTKDM4EALDH1A1
SCHEMBL8997153 0.68 CYP4A11 (0.36) TLR7MAPTTHRBMEN1KMT2A
SCHEMBL8997195 0.67 ATIC (0.35) TLR7MAPTTHRBTP53P2RX3
SCHEMBL9844745 0.67 MAPT (0.35) TLR7MAPTKDM4EALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed