SCHEMBL9440144

SCHEMBL9440144

O=C(O)c1c2n(c3cc(-c4ccncc4)c(F)cc3c1=O)CS2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.37
TOP2B Q02880 2/20 0.37
CYP3A4 P08684 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
PRKD3 O94806 1/20 0.35
PIM1 P11309 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
IRAK1 P51617 1/20 0.35
RPS6KA3 P51812 1/20 0.35
DYRK1A Q13627 1/20 0.35
PIM3 Q86V86 1/20 0.35
CSNK1G3 Q9Y6M4 1/20 0.35
MAPK14 Q16539 1/20 0.35
CALML3 P27482 1/20 0.33
ADH5 P11766 1/20 0.33
METAP2 P50579 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568448 0.90 PIM1 (0.37) AKR1C3AKR1C2PRKD3PIM1GSK3A
SCHEMBL9568451 0.87 PIM1 (0.37) PRKD3PIM1GSK3AGSK3BIRAK1
SCHEMBL9568301 0.84 PIM1 (0.35) PRKD3PIM1GSK3AGSK3BIRAK1
SCHEMBL9568435 0.84 PRKAB2 (0.36) PRKD3PIM1GSK3AGSK3BIRAK1
SCHEMBL8323537 0.82 PIM1 (0.41) TOP2ATOP2BPRKD3PIM1GSK3A
SCHEMBL9522528 0.78 PIM1 (0.39) PRKD3PIM1GSK3AGSK3BIRAK1
SCHEMBL9568395 0.76 KDM4E (0.44) CYP3A4
SCHEMBL9568459 0.73 PRKCZ (0.44)
SCHEMBL9523354 0.72 PRKD3 (0.48) TOP2ATOP2BPRKD3PIM1GSK3A
SCHEMBL9525097 0.72 PRKD3 (0.47) TOP2ATOP2BCYP3A4PRKD3PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6016678-A None JP disclosed
JP-H0616678-A QUINOLINECARBOXYLIC ACID DERIVATIVE NIPPON SHINYAKU CO LTD 1994-01-25 JP disclosed
JP-H00616678-A 0001-01-01 JP disclosed