SCHEMBL9444367

SCHEMBL9444367

COc1ccc(CCN2CCC(Cc3ccc(NS(C)(=O)=O)cc3)CC2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.61
HTR1A P08908 2/20 0.56
SLC6A4 P31645 1/20 0.56
LMNA P02545 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.48
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
EBP Q15125 1/20 0.47
SIGMAR1 Q99720 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9678100 0.86 KCNH2 (0.48) ABCB1HTR1ASLC6A4LMNAALDH1A1
SCHEMBL9447564 0.85 ABCB1 (0.45) ABCB1HTR1ASLC6A4ALDH1A1EBP
SCHEMBL9444495 0.84 KCNH2 (0.58) ABCB1SMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL9681410 0.83 ABCB1 (0.43) ABCB1HTR1ASLC6A4ALDH1A1HTT
Hydrochloric Acid SCHEMBL9444430 0.83 KCNH2 (0.59) ABCB1SMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL9041547 0.80 ABCB1 (0.43) ABCB1HTR1ASLC6A4ALDH1A1HTT
SCHEMBL10645360 0.80 KMT2A (0.54) ABCB1ALDH1A1MAPTRAB9AEBP
SCHEMBL9028157 0.79 OPRM1 (0.48) HTT
SCHEMBL9444543 0.77 KDM2B (0.60) LMNAALDH1A1MAPTHTT
SCHEMBL9444379 0.77 CCR3 (0.49) HTR1ASLC6A4ALDH1A1HTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0235752-B1 Piperidine derivative, pharmaceutical composition containing the same and use EISAI CO LTD (JP) 1993-11-18 EP disclosed
US-5179095-A Antiarrhythmia agents EISAI CO., LTD. (JP) 1993-01-12 US disclosed
US-5118689-A Antiarrhythmia agents EISAI CO., LTD. (JP) 1992-06-02 US disclosed
US-4996215-A Antiarrythmia agents EISAI CO., LTD. (JP) 1991-02-26 US disclosed
EP-0235752-A2 Piperidine derivative, pharmaceutical composition containing the same and use Eisai Co., Ltd. (JP) 1987-09-09 EP disclosed