SCHEMBL9446233

SCHEMBL9446233

Brc1ccc(N(Cc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.51
HDAC1 Q13547 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
TSHR P16473 3/20 0.47
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
KCNA3 P22001 1/20 0.45
CYP2C19 P33261 1/20 0.42
MAPK1 P28482 2/20 0.41
CYP1A2 P05177 1/20 0.41
ALDH1A1 P00352 3/20 0.41
PYCR1 P32322 2/20 0.40
CNR2 P34972 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6922536 0.94 HDAC1 (0.56) NR3C2HDAC1HDAC8HDAC6TSHR
SCHEMBL9446230 0.89 NR3C2 (0.59) NR3C2HDAC1HDAC8HDAC6TSHR
SCHEMBL6171116 0.87 CYP3A4 (0.46) NR3C2HDAC1HDAC8HDAC6TSHR
SCHEMBL28376324 0.87 ESR1 (0.50) HDAC1HDAC8HDAC6TSHRHTT
SCHEMBL918512 0.87 NR3C2 (0.56) NR3C2HDAC1HDAC8HDAC6TSHR
Bromide SCHEMBL4613403 0.84 NR3C2 (0.55) NR3C2HDAC1HDAC8HDAC6TSHR
SCHEMBL6927897 0.83 HDAC1 (0.48) NR3C2HDAC1HDAC8HDAC6TSHR
SCHEMBL1702260 0.83 NR3C2 (0.54) NR3C2HDAC1HDAC8HDAC6TSHR
Ethylene SCHEMBL11428459 0.82 NR3C2 (0.53) NR3C2HDAC1HDAC8HDAC6TSHR
SCHEMBL9215401 0.82 HDAC1 (0.60) NR3C2HDAC1HDAC8HDAC6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5196606-A Aromatic tertiary amines, enamines, deoxybenzoins and benzils HAY ALLAN S (CA) 1993-03-23 US disclosed
US-5117062-A Aromatic tertiary amines, enamines, deoxybenzoins and benzils HAY ALLAN S (CA) 1992-05-26 US disclosed
US-5011998-A Aromatic tertiary amines, enamines, deoxybenzoins and benzils HAY ALLAN S (CA) 1991-04-30 US disclosed