SCHEMBL9447116

SCHEMBL9447116

CCCCS(=O)(=O)Nc1ccc(Oc2cccc3cccnc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.52
TP53 P04637 1/20 0.48
HTT P42858 1/20 0.48
HPGD P15428 3/20 0.46
LMNA P02545 2/20 0.46
MRGPRX1 Q96LB2 1/20 0.46
GLO1 Q04760 3/20 0.45
KDM4E B2RXH2 4/20 0.44
MAPT P10636 4/20 0.44
ALDH1A1 P00352 4/20 0.44
FABP1 P07148 1/20 0.43
GAA P10253 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
SLC40A1 Q9NP59 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9446951 0.90 MAPT (0.46) ARHPGDLMNAMRGPRX1GLO1
SCHEMBL9446965 0.90 TP53 (0.46) TP53HTTLMNAGLO1KDM4E
SCHEMBL9446988 0.87 AR (0.48) ARTP53HTTHPGDLMNA
SCHEMBL9446997 0.84 AR (0.49) ARHPGDLMNAMRGPRX1KDM4E
SCHEMBL9447062 0.83 GLO1 (0.57) HTTMRGPRX1GLO1KDM4EALDH1A1
SCHEMBL8307237 0.81 AR (0.56) ARHTTHPGDLMNAMRGPRX1
SCHEMBL9447003 0.80 AR (0.52) ARHTTHPGDLMNAKDM4E
SCHEMBL9446959 0.80 AR (0.52) ARHTTHPGDLMNAMRGPRX1
SCHEMBL9447040 0.80 FABP1 (0.46) LMNAGLO1KDM4EMAPTFABP1
SCHEMBL9447167 0.80 AR (0.49) ARHPGDLMNAGLO1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202336-A Lipoxygenase inhibitors BAYER AKTIENGESELLSCHAFT (DE) 1993-04-13 US disclosed
US-5093340-A Lipoxygenase enzyme inhibitors, antithrombolytic agents BAYER AKTIENGESELLSCHAFT (DE) 1992-03-03 US disclosed
US-5070096-A ANTICOAGULANTS, LIPOXYGENASE INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 1991-12-03 US disclosed
EP-0261539-B1 SUBSTITUTED PHENYL-SULPHON AMIDES BAYER AG (DE) 1991-03-06 EP disclosed
EP-0261539-A2 Substituted phenyl-sulphon amides BAYER AG (DE) 1988-03-30 EP disclosed