SCHEMBL9447692

SCHEMBL9447692

Cc1c(CC(=O)O)c2cc(OCc3ccc4ccccc4n3)ccc2n1Cc1ccc(F)cc1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.64
CYP2C9 P11712 3/20 0.64
LMNA P02545 2/20 0.64
CYP1A2 P05177 2/20 0.64
TSHR P16473 2/20 0.64
CYP2C19 P33261 2/20 0.64
PMP22 Q01453 2/20 0.64
KDM4E B2RXH2 1/20 0.64
BLM P54132 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
PTGDR2 Q9Y5Y4 2/20 0.63
ALOX5AP P20292 9/20 0.61
PLA2G2A P14555 5/20 0.57
PLA2G1B P04054 1/20 0.57
PTGIR P43119 1/20 0.56
PTGDR Q13258 1/20 0.56
PTGS1 P23219 1/20 0.53
PTGS2 P35354 1/20 0.53
ALOX5 P09917 1/20 0.53
CYP2D6 P10635 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9146626 0.99 CYP3A4 (0.63) CYP3A4CYP2C9LMNACYP1A2TSHR
Water SCHEMBL9146635 0.99 CYP3A4 (0.63) CYP3A4CYP2C9LMNACYP1A2TSHR
SCHEMBL9680113 0.95 ALOX5AP (0.62) CYP3A4CYP2C9LMNACYP1A2TSHR
Water SCHEMBL9140717 0.94 ALOX5AP (0.61) CYP3A4CYP2C9LMNACYP1A2TSHR
Water SCHEMBL9140709 0.94 ALOX5AP (0.61) CYP3A4CYP2C9LMNACYP1A2TSHR
SCHEMBL9140666 0.94 PLA2G2A (0.65) CYP3A4CYP2C9LMNACYP1A2TSHR
SCHEMBL2746925 0.92 ALOX5AP (0.68) CYP3A4CYP2C9LMNACYP1A2TSHR
Hydrochloric Acid SCHEMBL9138311 0.92 ALOX5AP (0.67) CYP3A4CYP2C9LMNACYP1A2TSHR
SCHEMBL9138282 0.92 PLA2G2A (0.59) CYP3A4CYP2C9LMNACYP1A2TSHR
SCHEMBL9447721 0.92 PTGS2 (0.64) PTGDR2ALOX5APPLA2G2APLA2G1BPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229516-A Antiinflammatory agents, antiallergens and cytoprotective agents AMERICAN HOME PRODUCTS CORPORATION (US) 1993-07-20 US claimed
EP-0502106-A1 SUBSTITUTED INDOLE-, INDENE-, PYRANOINDOLE- AND TETRAHYDROCARBAZOLE- ALKANOIC ACID DERIVATIVES AS INHIBITORS OF PLA2 AND LIPOXYGENASE AMERICAN HOME PRODUCTS CORPORATION (US) 1992-09-09 EP claimed
WO-1991006537-A2 SUBSTITUTED INDOLE-, INDENE-, PYRANOINDOLE- AND TETRAHYDROCARBAZOLE- ALKANOIC ACID DERIVATIVES AS INHIBITORS OF PLA2 AND LIPOXYGENASE AMERICAN HOME PRODUCTS CORPORATION (US) 1991-05-16 WO claimed