SCHEMBL9448356

SCHEMBL9448356

NC(=O)c1cccc(OCC2CO2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.66
TP53 P04637 1/20 0.66
CYP3A4 P08684 1/20 0.66
TSHR P16473 1/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
HIF1A Q16665 1/20 0.66
TDP1 Q9NUW8 1/20 0.54
PARP1 P09874 3/20 0.51
PARP15 Q460N3 4/20 0.49
PARP10 Q53GL7 4/20 0.49
PARP2 Q9UGN5 3/20 0.49
TNKS O95271 1/20 0.49
PARP14 Q460N5 1/20 0.49
TNKS2 Q9H2K2 1/20 0.49
OPRK1 P41145 5/20 0.45
NR1H4 Q96RI1 1/20 0.44
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
KCNH2 Q12809 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208400 0.87 ALDH1A1 (0.68) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL19827992 0.87 ALDH1A1 (0.68) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL6915703 0.85 SMN1; SMN2 (0.66) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL6915699 0.85 SMN1; SMN2 (0.66) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL6915692 0.85 SMN1; SMN2 (0.66) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL19827996 0.85 ALDH1A1 (0.66) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL11198075 0.84 ALDH1A1 (0.64) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL32684970 0.83 SMN1; SMN2 (0.62) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2
SCHEMBL201939 0.82 PARP10 (0.67) PARP1PARP15PARP10PARP2TNKS
SCHEMBL4656658 0.81 PARP10 (0.66) ALDH1A1TP53CYP3A4TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5215738-A Used for destroying hypoxic tumor cells SRI INTERNATIONAL (US) 1993-06-01 US disclosed
US-5041653-A Antitumor agents SRI INTERNATIONAL (US) 1991-08-20 US disclosed
US-5032617-A Antitumor agents SRI INTERNATIONAL (US) 1991-07-16 US disclosed
US-4863903-A RENIN ENZYME INHIBITORS, HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1989-09-05 US disclosed
US-4719288-A HYPOTENSIVE CIBA-GEIGY CORPORATION (US) 1988-01-12 US disclosed
WO-1986006628-A1 BENZAMIDE AND NICOTINAMIDE RADIOSENSITIZERS SRI INTERNATIONAL (US) 1986-11-20 WO disclosed
US-4613676-A PEPTIDES CIBA-GEIGY CORPORATION (US) 1986-09-23 US disclosed