SCHEMBL9455447

SCHEMBL9455447

N#CC(Cl)(c1cccnc1)c1ccc(N)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.40
CYP3A4 P08684 5/20 0.36
CYP3A5 P20815 5/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.35
PSIP1 O75475 1/20 0.35
AXL P30530 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
ALDH1A1 P00352 1/20 0.34
ADORA2A P29274 1/20 0.33
CTSC P53634 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9787304 0.77 CYP3A4 (0.38) CYP3A4MEN1ALDH1A1
SCHEMBL9787321 0.75 CYP3A4 (0.43) CYP3A4POLBALDH1A1
SCHEMBL9455376 0.75 SYK (0.37) CYP3A4ALDH1A1
SCHEMBL5566635 0.73 CYP3A4 (0.70) CYP19A1CYP3A4CYP3A5
SCHEMBL9455534 0.70 KDM4E (0.45) CYP3A4MEN1ALDH1A1
SCHEMBL9455570 0.68 CASR (0.48) POLBMEN1ALDH1A1
SCHEMBL9455538 0.67 KIF11 (0.31) CYP3A4POLBMEN1ALDH1A1
SCHEMBL2819804 0.66 CYP3A4 (0.44) CYP3A4POLBMEN1ALDH1A1
SCHEMBL10421682 0.65 CYP3A4 (0.39) CYP3A4POLBMEN1ALDH1A1
SCHEMBL9770755 0.65 CYP3A4 (0.43) CYP19A1CYP3A4CYP3A5POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5196562-A Substituted 1,3,5-triazinetriones, for use against parasitic protozoa BAYER AKTIENGESELLSCHAFT (DE) 1993-03-23 US disclosed
US-4933341-A Substituted 1,3,5-triazinetriones, for use against parasitic protozoa BAYER AKTIENGESELLSCHAFT (DE) 1990-06-12 US disclosed
EP-0364765-A2 Substituted 1,3,5-triazinetriones, process for their preparation, and their use against parasitical protozoa BAYER AG (DE) 1990-04-25 EP disclosed