SCHEMBL9458046

SCHEMBL9458046

FC(F)(F)COc1cccc(I)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.49
MAPT P10636 4/20 0.46
ALDH1A1 P00352 3/20 0.46
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
CYP2C9 P11712 2/20 0.41
CYP17A1 P05093 1/20 0.41
CYP2C19 P33261 1/20 0.41
CETP P11597 1/20 0.40
HTT P42858 2/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
S1PR2 O95136 1/20 0.40
S1PR4 O95977 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10972329 0.86 MAPT (0.59) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL3923640 0.81 MAPT (0.50) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL28221173 0.78 MAPT (0.47) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL30167649 0.78 L3MBTL1 (0.55) MAPTALDH1A1HTTKDM4EKMT2A
SCHEMBL5843821 0.78 CETP (0.47) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL21246500 0.78 APP (0.42) ALDH1A1SMN1; SMN2APP
SCHEMBL24305918 0.77 MAPK1 (0.55) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL4348572 0.77 ACHE (0.50) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL1471132 0.77 MAOB (0.55) GPR3MAPTALDH1A1GRIN1GRIN2A
SCHEMBL10573493 0.77 MAPT (0.46) GPR3MAPTALDH1A1GRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed
EP-0409413-A2 Diaryl ether heterocycles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed