Phenyl Biguanide

Phenyl Biguanide

SCHEMBL9459112

C1CC1.N=C(N)NC(=N)Nc1ccccc1.N=C(N)NC(=N)Nc1ccccc1

nearest known ligand 0.45

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
TAS2R38 P59533 3/20 0.45
TP53 P04637 2/20 0.45
TSHR P16473 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TYR P14679 1/20 0.45
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
GLA P06280 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 4/20 0.40
MAPT P10636 1/20 0.40
GFER P55789 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
LMNA P02545 1/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenyl Biguanide SCHEMBL467623 0.94 ALDH1A1 (0.50) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL2721730 0.92 ALDH1A1 (0.48) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL28093786 0.92 ALDH1A1 (0.48) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL1989457 0.90 ALDH1A1 (0.47) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL27966288 0.90 POLB (0.42) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL16702225 0.89 GAA (0.48) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL1592736 0.87 MAPT (0.47) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL27966486 0.85 HSD17B10 (0.52) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL28429189 0.85 ACP1 (0.44) ALDH1A1TAS2R38TP53TSHRHSD17B10
Phenyl Biguanide SCHEMBL28014085 0.85 ALDH1A1 (0.43) ALDH1A1TAS2R38TP53TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0562668-A1 Monirritating antitartar and antiplaque oral compositions UNILEVER N.V. (NL) 1993-09-29 EP disclosed
US-5192533-A Hypophite-acrylic polymer CHESEBROUGH-POND'S USA CO., DIVISION OF CONOPCO, INC. (US) 1993-03-09 US disclosed
US-4886658-A MIXTURE OF MONOPEROXYPHTHALATE AND BISGUANID COMPOUND THE PROCTER & GAMBLE COMPANY (US) 1989-12-12 US disclosed
US-4157387-A Dentifrice composition containing an abrasive coated with a cationic water soluble polymer THE PROCTER & GAMBLE COMPANY (US) 1979-06-05 US disclosed
US-4110083-A HARD MINERAL PARTICLES COATED WITH A CATIONIC WATER-SOLUBLE POLYMER THE PROCTER & GAMBLE COMPANY (US) 1978-08-29 US disclosed
US-4025616-A Oral compositions for plaque, caries and calculus retardation with reduced staining tendencies THE PROCTER & GAMBLE COMPANY (US) 1977-05-24 US disclosed
US-3934002-A BIS-GUANIDE THE PROCTER & GAMBLE COMPANY (US) 1976-01-20 US disclosed