SCHEMBL9459488

SCHEMBL9459488

O=S(=O)(c1ccc(Br)cc1)c1cccc(F)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.53
HTR2B P41595 1/20 0.53
HTR2A P28223 3/20 0.49
ABCC9 O60706 1/20 0.48
ABCC8 Q09428 1/20 0.48
KCNJ11 Q14654 1/20 0.48
KCNJ8 Q15842 1/20 0.48
ALDH1A1 P00352 1/20 0.48
KCNH2 Q12809 2/20 0.45
HTR6 P50406 5/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MAPT P10636 1/20 0.45
NFE2L2 Q16236 2/20 0.43
LMNA P02545 1/20 0.42
NAMPT P43490 2/20 0.42
GAA P10253 2/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9460224 0.87 HTR2C (0.50) HTR2CHTR2BHTR2AABCC9ABCC8
SCHEMBL7182433 0.86 HTR2A (0.60) HTR2CHTR2BHTR2AABCC9ABCC8
SCHEMBL18187421 0.86 ALDH1A1 (0.58) ALDH1A1HTR6SMN1; SMN2MAPTLMNA
SCHEMBL775608 0.86 HTR2C (0.59) HTR2CHTR2BHTR2AABCC9ABCC8
SCHEMBL777135 0.84 HTR6 (0.61) HTR2CHTR2BHTR2AABCC9ABCC8
SCHEMBL28582400 0.82 ALDH1A1 (0.59) HTR2CHTR2BALDH1A1HTR6SMN1; SMN2
SCHEMBL15239367 0.82 ALDH1A1 (0.51) ALDH1A1HTR6SMN1; SMN2MAPTLMNA
SCHEMBL9459975 0.81 EGFR (0.48) HTR2CHTR2BHTR2AALDH1A1KCNH2
SCHEMBL24720985 0.81 GAA (0.59) HTR2CHTR2BHTR2AABCC9ABCC8
SCHEMBL3446114 0.81 ALDH1A1 (0.59) HTR2CHTR2BHTR2AABCC9ABCC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5185454-A Reacting aryl bromide with acetylene in presence of palladium catalyst and nitrogen-containing heterocyclic base BAYER AKTIENGESELLSCHAFT (DE) 1993-02-09 US disclosed