SCHEMBL9466779

SCHEMBL9466779

O=C(CCCN1C=CC(C2=CCC=CC2)=CC1)c1ccncc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.33
HTR2C P28335 4/20 0.33
SLC6A4 P31645 1/20 0.33
HRH1 P35367 2/20 0.32
HRH2 P25021 1/20 0.32
DRD2 P14416 5/20 0.32
HTR1A P08908 4/20 0.32
DRD4 P21917 4/20 0.32
DRD3 P35462 4/20 0.32
ADRA2C P18825 1/20 0.32
CTNNB1 P35222 1/20 0.31
WNT3A P56704 1/20 0.31
HTR7 P34969 3/20 0.31
TMEM97 Q5BJF2 2/20 0.30
SIGMAR1 Q99720 2/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9473855 0.81 SIGMAR1 (0.36) HRH1SIGMAR1CYP1A2CYP3A4
SCHEMBL9466840 0.80 SIGMAR1 (0.40) SLC6A4HRH1DRD4SIGMAR1CYP1A2
SCHEMBL9467956 0.78
SCHEMBL8908199 0.74 DRD2 (0.42) DRD2DRD4DRD3
SCHEMBL11828755 0.71
SCHEMBL9826487 0.69 KCNA3 (0.44) HTR2ADRD2DRD3HTR7
SCHEMBL8906856 0.69 DRD2 (0.46) DRD2DRD4DRD3CYP1A2CYP3A4
SCHEMBL9874339 0.65
SCHEMBL8906800 0.64 DRD2 (0.46) DRD2DRD4DRD3
Bromide SCHEMBL29288531 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed