SCHEMBL9826487

SCHEMBL9826487

C1=CCC(C2=CCN(CCCOc3cccc4cnccc34)C=C2)=CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.44
HRH3 Q9Y5N1 4/20 0.34
MAPT P10636 2/20 0.34
DRD3 P35462 2/20 0.34
METAP2 P50579 1/20 0.33
NR3C1 P04150 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
HTR1B P28222 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
HTR7 P34969 1/20 0.31
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9826733 0.99 KCNA3 (0.43) KCNA3HRH3MAPTDRD3METAP2
SCHEMBL9825711 0.80 HTR1A (0.43) MAPTDRD3HTR1BDRD2
SCHEMBL9473855 0.73 SIGMAR1 (0.36) HRH3TDP1
SCHEMBL9466840 0.73 SIGMAR1 (0.40) HRH3TDP1
SCHEMBL9826279 0.72 CYP2D6 (0.39) HRH3MAPTDRD3
Hydrochloric Acid SCHEMBL9719843 0.70 HTR3A (0.32)
SCHEMBL9466779 0.69 HTR2A (0.33) DRD3DRD2HTR2AHTR7
Water SCHEMBL9825376 0.69 LTA4H (0.37) DRD3DRD2
SCHEMBL8906856 0.68 DRD2 (0.46) DRD3DRD2
SCHEMBL10576049 0.67 KCNA3 (0.69) KCNA3MAPTNR3C1TDP1HTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237781-B1 PHENYL AND HETEROCYCLIC TETRAHYDROPYRIDYL AND PIPERAZINYL ALKOXY-BENZHETEROCYCLIC COMPOUNDS AS ANTIPSYCHOTIC AGENTS WARNER-LAMBERT COMPANY (US) 1991-04-24 EP claimed
US-4704390-A SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1987-11-03 US claimed
EP-0237781-A2 Phenyl and heterocyclic tetrahydropyridyl and piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents WARNER-LAMBERT COMPANY (US) 1987-09-23 EP claimed
EP-0237781-B1 PHENYL AND HETEROCYCLIC TETRAHYDROPYRIDYL AND PIPERAZINYL ALKOXY-BENZHETEROCYCLIC COMPOUNDS AS ANTIPSYCHOTIC AGENTS WARNER-LAMBERT COMPANY (US) 1991-04-24 EP disclosed
US-4803203-A SCHIZOPHRENIA, NEUOLEPTIC AGENTS WARNER-LAMBERT COMPANY (US) 1989-02-07 US disclosed
US-4704390-A SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1987-11-03 US disclosed
EP-0237781-A2 Phenyl and heterocyclic tetrahydropyridyl and piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents WARNER-LAMBERT COMPANY (US) 1987-09-23 EP disclosed