SCHEMBL9468664

SCHEMBL9468664

CC/C(=C\N(C)C)C(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.58
ALDH1A1 P00352 2/20 0.56
POLB P06746 1/20 0.49
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
SRD5A2 P31213 1/20 0.43
MAOB P27338 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CCR2 P41597 1/20 0.42
OPRM1 P35372 1/20 0.42
OPRL1 P41146 1/20 0.42
P2RX1 P51575 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9468665 1.00 CES2 (0.58) CES2ALDH1A1POLBTAS1R3TAS1R1
SCHEMBL9874158 0.83 CYP11B1 (0.54) CES2SRD5A2MAOB
SCHEMBL11465984 0.82 CES2 (0.63) CES2ALDH1A1POLBNPSR1SRD5A2
SCHEMBL11465983 0.82 CES2 (0.63) CES2ALDH1A1POLBNPSR1SRD5A2
SCHEMBL9160769 0.81 CES2 (0.58) CES2ALDH1A1POLBNPSR1SRD5A2
SCHEMBL11376363 0.79 CES2 (0.51) CES2ALDH1A1POLBTAS1R3TAS1R1
SCHEMBL3544067 0.79 CES2 (0.51) CES2ALDH1A1POLBTAS1R3TAS1R1
SCHEMBL13729327 0.78 CES2 (0.53) CES2ALDH1A1MEN1KMT2A
SCHEMBL9159447 0.77 CES2 (0.56) CES2ALDH1A1POLBNPSR1SRD5A2
SCHEMBL9159450 0.77 CES2 (0.56) CES2ALDH1A1POLBNPSR1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5219857-A Method of treating cognitive and related neural behavioral problems AMERICAN CYANAMID COMPANY (US) 1993-06-15 US disclosed
US-5126340-A Antidepressants AMERICAN CYANAMID COMPANY (US) 1992-06-30 US disclosed
US-4963553-A TREATING COGNITIVE AND NEURAL BEHAVIORAL PROBLEMS IN MAMMALS AMERICAN CYANAMID CO. (US) 1990-10-16 US disclosed
EP-0264773-A1 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1988-04-27 EP disclosed