SCHEMBL947083

SCHEMBL947083

COc1c(C)cc(C2(c3cccc(Br)c3)N=C(C)C(=S)N2)cc1C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
RXFP1 Q9HBX9 1/20 0.32
KCNH2 Q12809 1/20 0.32
CHRNA1 P02708 1/20 0.30
CHRNG P07510 1/20 0.30
CHRNB1 P11230 1/20 0.30
CHRNB2 P17787 1/20 0.30
SLC6A2 P23975 1/20 0.30
CHRNB4 P30926 1/20 0.30
SLC6A4 P31645 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30
SLC6A3 Q01959 1/20 0.30
CHRND Q07001 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920536 0.87 BACE1 (0.39) BACE1BACE2
SCHEMBL932469 0.86 BACE1 (0.31) BACE1
SCHEMBL944383 0.85
SCHEMBL944396 0.83 NCOA1 (0.33) RXFP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL945865 0.80 ALDH1A1 (0.35) BACE1BACE2RXFP1
SCHEMBL947897 0.77 BACE1 (0.31) BACE1BACE2
SCHEMBL946379 0.72
SCHEMBL932204 0.71 BACE1 (0.67) BACE1BACE2KCNH2
SCHEMBL943316 0.69 ALDH1A1 (0.34) BACE1RXFP1CHRNA1CHRNGCHRNB1
SCHEMBL945249 0.68 CHRNA1 (0.37) BACE1CHRNA1CHRNGCHRNB1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed