SCHEMBL9475423

SCHEMBL9475423

COc1ccc(CSC2=NC(C)=C(C(=O)O)C(c3cccc4nonc34)N2C(=O)O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
HTT P42858 3/20 0.39
RECQL P46063 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
TP53 P04637 1/20 0.37
KMT2A Q03164 5/20 0.37
FFAR1 O14842 1/20 0.36
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
MLNR O43193 1/20 0.35
NR1I2 O75469 1/20 0.35
ABCB11 O95342 1/20 0.35
NR3C1 P04150 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CYP2C8 P10632 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9475146 0.84 PTGDR2 (0.42) ALDH1A1PTGDR2TP53FFAR1MAPT
SCHEMBL9476368 0.83 TP53 (0.40) ALDH1A1PTGDR2TP53KMT2AFFAR1
SCHEMBL9475728 0.83 ABL1 (0.41) ALDH1A1PTGDR2KMT2AFFAR1MAPT
SCHEMBL9476156 0.82 FFAR1 (0.38) PTGDR2FFAR1MAPTGAACACNA1C
SCHEMBL9476315 0.82 MAPT (0.41) ALDH1A1HTTPTGDR2KMT2AFFAR1
SCHEMBL9476961 0.80 FFAR1 (0.44) ALDH1A1HTTPTGDR2TP53KMT2A
SCHEMBL9476024 0.80 ALDH1A1 (0.41) ALDH1A1PTGDR2KMT2AFFAR1GAA
SCHEMBL9475639 0.79 TP53 (0.40) ALDH1A1HTTPTGDR2TP53KMT2A
SCHEMBL9476282 0.79 SMN1; SMN2 (0.41) ALDH1A1HTTPTGDR2KMT2AMAPT
SCHEMBL9476099 0.79 POLB (0.40) PTGDR2TP53FFAR1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202330-A Hypotensive and cardiovascular agent, reduces blood pressure in mammals E. R. SQUIBB & SONS, INC. (US) 1993-04-13 US disclosed
EP-0204317-A2 2-Thio or oxo-4-aryl or heterocyclo-1,5(2H)-pyrimidinedicarboxylic acid diesters and 3-acyl-5-pyrimidinecarboxylic acids and esters E.R. Squibb & Sons, Inc. (US) 1986-12-10 EP disclosed