SCHEMBL9475577

SCHEMBL9475577

NC(=O)c1nnn(Cc2ccccc2F)c1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.52
MAPT P10636 3/20 0.49
TP53 P04637 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
CYP1A2 P05177 1/20 0.47
GALR3 O60755 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
NR2F2 P24468 1/20 0.46
HIF1A Q16665 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
GRM2 Q14416 1/20 0.45
TSHR P16473 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ATM Q13315 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857450 0.86 GRM2 (0.45) HPGDMAPTALDH1A1MEN1KMT2A
SCHEMBL8008741 0.85 MAPT (0.57) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL9476992 0.84 CA5A (0.53) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL9478376 0.83 NPC1 (0.56) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL9477082 0.83 NPSR1 (0.65) HPGDMAPTALDH1A1HTTNPSR1
SCHEMBL10669535 0.83 HPGD (0.52) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL10666397 0.83 HPGD (0.49) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL19743797 0.80 HPGD (0.49) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL19743408 0.80 HPGD (0.52) HPGDMAPTTP53ALDH1A1HTT
SCHEMBL11245223 0.80 HPGD (0.80) HPGDMAPTTP53HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0114347-A2 Aralkyl-triazole compounds CIBA-GEIGY AG (CH) 1984-08-01 EP claimed
US-5204353-A 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith CIBA-GEIGY CORPORATION (US) 1993-04-20 US disclosed
EP-0288431-B1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1992-08-19 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0288431-A1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1988-10-26 EP disclosed
EP-0114347-A2 Aralkyl-triazole compounds CIBA-GEIGY AG (CH) 1984-08-01 EP disclosed