SCHEMBL9475648

SCHEMBL9475648

CC1CN(c2c(F)cc3c(=O)c(C(=O)O)cn(C4CC4)c3c2C#N)CCN1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.74
ALDH1A1 P00352 7/20 0.74
KDM4E B2RXH2 7/20 0.74
HPGD P15428 7/20 0.74
HSD17B10 Q99714 5/20 0.74
POLB P06746 3/20 0.74
OPRM1 P35372 2/20 0.74
PRKD3 O94806 1/20 0.74
ALOX15 P16050 1/20 0.74
CLK2 P49760 1/20 0.74
CLK4 Q9HAZ1 1/20 0.74
TDP1 Q9NUW8 1/20 0.74
PMP22 Q01453 1/20 0.60
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
OPRD1 P41143 1/20 0.54
HRH3 Q9Y5N1 1/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
LMNA P02545 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12917214 0.90 MEN1 (0.62) KCNH2ALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL967940 0.89 MEN1 (0.61) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL29593740 0.89 ALDH1A1 (0.81) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6783172 0.89 ALDH1A1 (0.81) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10697767 0.89 KDM4E (0.61) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9474947 0.88 TOP2A (0.61) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9260082 0.88 KCNH2 (0.69) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9475858 0.88 KDM4E (0.57) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3957125 0.87 ALDH1A1 (0.79) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9792010 0.87 KCNH2 (0.79) KCNH2ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5190955-A Bactericides, effective against antibiotic resistant germs BAYER AKTIENGESELLSCHAFT (DE) 1993-03-02 US disclosed
US-5051418-A Antibacterial 8-cyano-1-cyclopropyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1991-09-24 US disclosed
US-4908366-A Bactericides BAYER AKTIENGESELLSCHAFT (DE) 1990-03-13 US disclosed
EP-0276700-A1 8-Cyano-1-cyclopropyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids, process for their preparation, and antibacterial agents containing them BAYER AG (DE) 1988-08-03 EP disclosed