SCHEMBL9792010

SCHEMBL9792010

Cc1c(N2CCNC(C)C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.79
ALDH1A1 P00352 7/20 0.79
KDM4E B2RXH2 6/20 0.79
HPGD P15428 6/20 0.79
HSD17B10 Q99714 5/20 0.79
POLB P06746 3/20 0.79
OPRM1 P35372 2/20 0.79
PRKD3 O94806 1/20 0.79
ALOX15 P16050 1/20 0.79
CLK2 P49760 1/20 0.79
CLK4 Q9HAZ1 1/20 0.79
TDP1 Q9NUW8 1/20 0.79
PMP22 Q01453 1/20 0.64
HRH3 Q9Y5N1 1/20 0.61
CHRM2 P08172 1/20 0.58
CHRM1 P11229 1/20 0.58
OPRD1 P41143 1/20 0.58
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
LMNA P02545 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29593740 0.92 ALDH1A1 (0.81) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6783172 0.92 ALDH1A1 (0.81) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3957125 0.91 ALDH1A1 (0.79) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8433684 0.90 ALDH1A1 (0.77) KCNH2ALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL10352018 0.89 ALDH1A1 (0.76) KCNH2ALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL10914782 0.89 ALDH1A1 (0.76) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9485535 0.89 ALDH1A1 (0.76) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9676493 0.88 KCNH2 (0.68) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9479924 0.88 ALDH1A1 (0.75) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10573958 0.88 ALDH1A1 (0.75) KCNH2ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4874764-A ANTIMICROBIALS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-10-17 US claimed
JP-3081224-A None JP disclosed
JP-H0381224-A THERAPEUTIC AGENT FOR LEPROSY OTSUKA PHARMACEUT CO LTD 1991-04-05 JP disclosed
US-4880806-A BACTERICIDES OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-11-14 US disclosed
US-4874764-A ANTIMICROBIALS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-10-17 US disclosed