SCHEMBL947597

SCHEMBL947597

COC(=O)CC1c2[nH]c3ccc(OCc4ccc(C(F)(F)F)cc4)cc3c2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.55
TRPV1 Q8NER1 1/20 0.45
HDAC1 Q13547 2/20 0.44
S1PR4 O95977 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
S1PR5 Q9H228 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL948110 0.89 S1PR1 (0.59) S1PR1S1PR4ADORA3S1PR5
SCHEMBL944763 0.83 TRPV1 (0.50) TRPV1
SCHEMBL950202 0.82 S1PR1 (0.60) S1PR1S1PR4S1PR5
SCHEMBL949739 0.82 S1PR1 (0.53) S1PR1S1PR4ADORA3S1PR5
SCHEMBL945721 0.81 MAPKAPK2 (0.56) S1PR1
Hydrochloric Acid SCHEMBL949245 0.79 S1PR1 (0.81) S1PR1S1PR4S1PR5
SCHEMBL947736 0.78 SLC6A4 (0.42) TRPV1
SCHEMBL945300 0.77 S1PR1 (0.75) S1PR1S1PR4ADORA3S1PR5
SCHEMBL946705 0.77 S1PR1 (0.68) S1PR1S1PR4ADORA3S1PR5
SCHEMBL951334 0.77 S1PR1 (0.60) S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed