SCHEMBL950202

SCHEMBL950202

COC(=O)CC1c2[nH]c3ccc(OCc4ccc(OC(C)C)c(C#N)c4)cc3c2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.60
S1PR5 Q9H228 2/20 0.46
S1PR4 O95977 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL947597 0.82 S1PR1 (0.55) S1PR1S1PR5S1PR4
SCHEMBL948110 0.81 S1PR1 (0.59) S1PR1S1PR5S1PR4
SCHEMBL947736 0.80 SLC6A4 (0.42)
Trifluoroacetic Acid SCHEMBL948308 0.78 S1PR1 (0.80) S1PR1S1PR5S1PR4
SCHEMBL944763 0.78 TRPV1 (0.50)
SCHEMBL1918221 0.76 S1PR1 (0.83) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL1918217 0.76 S1PR1 (0.83) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL30534223 0.76 S1PR1 (0.83) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL30534220 0.76 S1PR1 (0.83) S1PR1S1PR5S1PR4CYP2C9
SCHEMBL30534221 0.76 S1PR1 (0.83) S1PR1S1PR5S1PR4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed