SCHEMBL948110

SCHEMBL948110

COC(=O)CC1c2[nH]c3ccc(OCc4ccc(Cl)c(C(F)(F)F)c4)cc3c2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.59
S1PR4 O95977 2/20 0.47
S1PR5 Q9H228 2/20 0.47
ADORA3 P0DMS8 1/20 0.47
S1PR2 O95136 1/20 0.45
S1PR3 Q99500 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL947597 0.89 S1PR1 (0.55) S1PR1S1PR4S1PR5ADORA3
SCHEMBL951334 0.82 S1PR1 (0.60) S1PR1
SCHEMBL945075 0.81 S1PR1 (0.53) S1PR1S1PR4S1PR5ADORA3S1PR2
SCHEMBL950202 0.81 S1PR1 (0.60) S1PR1S1PR4S1PR5
SCHEMBL949534 0.81 S1PR1 (0.84) S1PR1S1PR4S1PR5S1PR2S1PR3
SCHEMBL945300 0.80 S1PR1 (0.75) S1PR1S1PR4S1PR5ADORA3S1PR2
SCHEMBL946705 0.80 S1PR1 (0.68) S1PR1S1PR4S1PR5ADORA3S1PR2
SCHEMBL944763 0.80 TRPV1 (0.50)
SCHEMBL949739 0.78 S1PR1 (0.53) S1PR1S1PR4S1PR5ADORA3
SCHEMBL946551 0.77 S1PR1 (0.53) S1PR1S1PR4S1PR5ADORA3S1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed