SCHEMBL9475989

SCHEMBL9475989

CN1CCC(C2=NC(C)(C)Oc3ccc(C#N)cc32)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 7/20 0.37
ABCC9 O60706 4/20 0.37
ABCC8 Q09428 2/20 0.37
KCNJ11 Q14654 2/20 0.37
KCNJ8 Q15842 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
LMNA P02545 1/20 0.37
BACE1 P56817 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HTR2A P28223 1/20 0.35
MAP3K5 Q99683 1/20 0.35
MALT1 Q9UDY8 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846798 0.74 PDE4A (0.39) ABCB1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9372531 0.70 ABCC9 (0.47) ABCB1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9375925 0.69 ABCC9 (0.44) ABCB1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9372439 0.69 ABCC9 (0.39) ABCB1ABCC9BACE1KDM4EMALT1
SCHEMBL9375996 0.69 ABCB1 (0.36) ABCB1ABCC9CYP1A2CYP2D6CYP2C19
SCHEMBL9372094 0.67 ABCC9 (0.36) ABCB1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9371935 0.67 ABCC9 (0.38) ABCB1ABCC9BACE1MAP3K5MALT1
SCHEMBL9377494 0.66 ABCC9 (0.38) ABCB1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9373199 0.66 ABCC9 (0.36) ABCB1ABCC9BACE1MALT1PDE4A
SCHEMBL9375563 0.66 ABCC9 (0.35) ABCB1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477789-A1 1,3-Benzoxazine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-01 EP claimed
US-5270308-A Hypotensives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-14 US disclosed
EP-0477789-A1 1,3-Benzoxazine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1992-04-01 EP disclosed