SCHEMBL9476396

SCHEMBL9476396

CNc1ncnc2c1nnn2Cc1ccccc1F

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.67
PKM P14618 3/20 0.65
POLB P06746 1/20 0.65
PDE4A P27815 3/20 0.65
PDE4B Q07343 3/20 0.65
PDE4C Q08493 3/20 0.65
PDE4D Q08499 3/20 0.65
PDE5A O76074 2/20 0.65
PDE1A P54750 2/20 0.65
PDE1B Q01064 2/20 0.65
PDE3B Q13370 2/20 0.65
PDE1C Q14123 2/20 0.65
PDE3A Q14432 2/20 0.65
LMNA P02545 3/20 0.57
MAPK1 P28482 2/20 0.55
TSHR P16473 2/20 0.55
HTT P42858 2/20 0.55
KDM4E B2RXH2 1/20 0.55
HSD17B10 Q99714 1/20 0.55
HPGD P15428 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9475021 0.86 ALDH1A1 (0.58) ALDH1A1PKMPOLBPDE4APDE4B
SCHEMBL9476085 0.86 ALDH1A1 (0.56) ALDH1A1PKMLMNAMAPK1TSHR
SCHEMBL9476378 0.85 ALDH1A1 (0.74) ALDH1A1PKMLMNAMAPK1TSHR
SCHEMBL9476453 0.85 ALDH1A1 (0.61) ALDH1A1PKMPOLBLMNAMAPK1
SCHEMBL9477074 0.84 ALDH1A1 (0.52) ALDH1A1PKMPOLBLMNAMAPK1
SCHEMBL9476430 0.82 ALDH1A1 (0.52) ALDH1A1PKMLMNAMAPK1TSHR
SCHEMBL9476117 0.81 ALDH1A1 (0.74) ALDH1A1POLBPDE4APDE4BPDE4C
SCHEMBL9475598 0.81 ALDH1A1 (0.61) ALDH1A1PKMPOLBLMNATSHR
SCHEMBL9475889 0.81 ALDH1A1 (0.61) ALDH1A1PKMPOLBLMNAMAPK1
SCHEMBL9475437 0.81 ADORA3 (0.61) ALDH1A1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288431-B1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1992-08-19 EP claimed
EP-0288431-A1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1988-10-26 EP claimed
US-5204353-A 3-benzyl-3H-1,2,3-triazolo[4,5-d]pyrimidines, compositions thereof, and method of treating epilepsy therewith CIBA-GEIGY CORPORATION (US) 1993-04-20 US disclosed
EP-0288431-B1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1992-08-19 EP disclosed
EP-0288431-A1 3H-1,2,3-triazolo[4,5-d]pyrimidines CIBA-GEIGY AG (CH) 1988-10-26 EP disclosed