Avarol

Avarol

SCHEMBL9477102

CC1=CCC[C@H]2[C@](C)(Cc3cc(O)ccc3O)[C@@H](C)CC[C@]12C.Oc1ccc(O)cc1

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 11/20 0.98
PTGS2 P35354 3/20 0.98
CETP P11597 1/20 0.98
PTPN6 P29350 3/20 0.61
ACLY P53396 3/20 0.61
IGF1R P08069 2/20 0.58
SRC P12931 2/20 0.58
AXL P30530 2/20 0.58
KDR P35968 2/20 0.58
PTK2 Q05397 2/20 0.58
ALK Q9UM73 2/20 0.58
NUAK1 O60285 1/20 0.58
MET P08581 1/20 0.58
PIM1 P11309 1/20 0.58
AKT1 P31749 1/20 0.58
NEK2 P51955 1/20 0.58
PLK1 P53350 1/20 0.58
AURKB Q96GD4 1/20 0.58
NEK6 Q9HC98 1/20 0.58
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Avarol SCHEMBL186460 0.99 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL21397196 0.99 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL31517137 0.99 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL10402772 0.99 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL9477704 0.96 PTPN1 (0.94) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL9478364 0.88 PTPN1 (0.80) PTPN1PTGS2CETPPTPN6ACLY
Avarone SCHEMBL5806251 0.87 PTPN1 (0.77) PTPN1PTGS2CETPPTPN6ACLY
SCHEMBL31536047 0.83 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
SCHEMBL31536088 0.80 PTPN1 (0.68) PTPN1PTGS2CETPPTPN6ACLY
SCHEMBL9478317 0.79 PTPN1 (0.78) PTPN1PTGS2CETPPTPN6ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5180748-A Antitumor agents MERZ+CO. GMBH & CO. (DE) 1993-01-19 US disclosed
US-5082865-A Avarol and its production and use as an antitumor agent (I) MUELLER WERNER E G (DE) 1992-01-21 US disclosed
US-4946869-A IN THE FORMS OF TABLETS, CAPSULES, ELIXIRS, SUPPOSITORIES OR STERILE INJECTABLE SOLUTIONS MERZ AND CO. GMBH & CO. (DE) 1990-08-07 US disclosed