Avarol

Avarol

SCHEMBL186460

CC1=CCC[C@H]2[C@](C)(Cc3cc(O)ccc3O)[C@@H](C)CC[C@]12C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 11/20 1.00
PTGS2 P35354 3/20 1.00
CETP P11597 1/20 1.00
PTPN6 P29350 3/20 0.62
ACLY P53396 3/20 0.62
IGF1R P08069 2/20 0.59
SRC P12931 2/20 0.59
AXL P30530 2/20 0.59
KDR P35968 2/20 0.59
PTK2 Q05397 2/20 0.59
ALK Q9UM73 2/20 0.59
NUAK1 O60285 1/20 0.59
MET P08581 1/20 0.59
PIM1 P11309 1/20 0.59
AKT1 P31749 1/20 0.59
NEK2 P51955 1/20 0.59
PLK1 P53350 1/20 0.59
AURKB Q96GD4 1/20 0.59
NEK6 Q9HC98 1/20 0.59
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Avarol SCHEMBL10402772 1.00 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL21397196 1.00 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL31517137 1.00 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL9477102 0.99 PTPN1 (0.98) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL9477704 0.97 PTPN1 (0.94) PTPN1PTGS2CETPPTPN6ACLY
Avarol SCHEMBL9478364 0.89 PTPN1 (0.80) PTPN1PTGS2CETPPTPN6ACLY
Avarone SCHEMBL5806251 0.88 PTPN1 (0.77) PTPN1PTGS2CETPPTPN6ACLY
SCHEMBL31536047 0.84 PTPN1 (1.00) PTPN1PTGS2CETPPTPN6ACLY
SCHEMBL31536088 0.81 PTPN1 (0.68) PTPN1PTGS2CETPPTPN6ACLY
SCHEMBL9478317 0.80 PTPN1 (0.78) PTPN1PTGS2CETPPTPN6ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1192 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026090160-A2 CD4-TARGETED IL-15 MOLECULES AND METHODS OF USE GILEAD SCIENCES, INC. (US) 2026-04-30 WO claimed
US-20250122146-A1 COMPOUNDS FOR REDUCING NEUROINFLAMMATION THE SCRIPPS RESEARCH INSTITUTE 2025-04-17 US claimed
CN-110678432-B Composition for completely or partially replacing ball clay in ceramic and preparation method and application thereof 活性矿物国际有限公司 2022-06-07 CN claimed
CN-110678432-A Composition for completely or partially replacing ball clay in ceramic and preparation method and application thereof 活性矿物国际有限公司 2020-01-10 CN claimed
JP-2011528275-A 2011-11-17 JP claimed
EP-2313122-A1 DRUG DELIVERY MEDICAL DEVICE Micell Technologies, Inc. (US) 2011-04-27 EP claimed
WO-2010009335-A1 DRUG DELIVERY MEDICAL DEVICE MICELL TECHNOLOGIES, INC. (US) 2010-01-21 WO claimed
US-20090054369-A1 PHARMACEUTICAL COMPOSITIONS OF SILICON-CONTAINING SUBSTITUTED ADENOSINE NUCLEOSIDE AMIDE ANALOGS RND PHARMACEUTICALS, INC. (US) 2009-02-26 US claimed
EP-1919929-A4 PHARMACEUTICAL COMPOSITIONS OF SILICON-CONTAINING SUBSTITUTED ADENOSINE NUCLEOSIDE AMIDE ANALOGS RND PHARMACEUTICALS INC (US) 2008-08-06 EP claimed
EP-1919929-A2 PHARMACEUTICAL COMPOSITIONS OF SILICON-CONTAINING SUBSTITUTED ADENOSINE NUCLEOSIDE AMIDE ANALOGS RND Pharmaceuticals, Inc. (US) 2008-05-14 EP claimed
EP-1391197-A1 Process for preparation of compositions with a high content in avarol and their use KliniPharm GmbH (DE) 2004-02-25 EP claimed
US-6075057-A INHIBITORS OF ALPHA-GLUCOSIDASE AND ALPHA-MANNOSIDASE; TREATMENT OF RETROVIRAL INFECTION-ASSOCIATED SYNDROMES, SUCH AS AIDS THE UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2000-06-13 US claimed
EP-0393575-B1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent SEARLE & CO (US) 1994-03-16 EP claimed
US-5082865-A Avarol and its production and use as an antitumor agent (I) MUELLER WERNER E G (DE) 1992-01-21 US claimed
EP-0393575-A1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent G.D. Searle & Co. (US) 1990-10-24 EP claimed
US-4946869-A IN THE FORMS OF TABLETS, CAPSULES, ELIXIRS, SUPPOSITORIES OR STERILE INJECTABLE SOLUTIONS MERZ AND CO. GMBH & CO. (DE) 1990-08-07 US claimed
US-4939178-A Use of avarol for the control of adult T-cell leukemia/lymphoma MERZ + CO. GMBH & CO. (DE) 1990-07-03 US claimed
US-4939177-A Use of avarol for the control of AIDS and ARC MERZ + CO. GMBH & CO. (DE) 1990-07-03 US claimed
EP-0252305-A2 Use of avarone and avarol and derivatives thereof for the preparation of a pharmaceutical composition for the control of adult T-cell leukemia/lymphoma Merz & Co. GmbH & Co. (DE) 1988-01-13 EP claimed
EP-0252304-A2 Use of avarone and avarol and derivatives thereof for the preparation of a pharmaceutical composition for the control of AIDS and ARC Merz & Co. GmbH & Co. (DE) 1988-01-13 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250122146-A1 COMPOUNDS FOR REDUCING NEUROINFLAMMATION HSF1, HSPA2, KEAP1 PTPN1 3982/4885PTGS2 267/4885CETP 4053/4885
US-20090054369-A1 PHARMACEUTICAL COMPOSITIONS OF SILICON-CONTAINING SUBSTITUTED ADENOSINE NUCLEOSIDE AMIDE ANALOGS SI, SLC29A2, SLC29A1 PTPN1 3857/4885PTGS2 2129/4885CETP 1987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.