SCHEMBL9480993

SCHEMBL9480993

CC1(C(=O)O)NCCc2c1[nH]c1ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.52
OPRM1 P35372 5/20 0.51
OPRL1 P41146 3/20 0.51
OGFRL1 Q5TC84 3/20 0.51
KMT2A Q03164 4/20 0.51
KDM4E B2RXH2 3/20 0.49
MAPKAPK2 P49137 1/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
MEN1 O00255 3/20 0.44
MAPT P10636 3/20 0.43
HTR5A P47898 1/20 0.43
NISCH Q9Y2I1 1/20 0.43
NR2E1 Q9Y466 1/20 0.43
CRHBP P24387 1/20 0.42
MAPK1 P28482 1/20 0.42
CRHR2 Q13324 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11318061 0.85 LMNA (0.49) LMNAOPRM1OPRL1OGFRL1KMT2A
SCHEMBL6238822 0.85 KMT2A (0.51) LMNAOPRM1OPRL1OGFRL1KMT2A
SCHEMBL31171169 0.83 MAPKAPK2 (0.49) OPRM1OGFRL1KDM4EMAPKAPK2ALDH1A1
SCHEMBL9685713 0.82 KMT2A (0.62) LMNAOPRM1OPRL1OGFRL1KMT2A
SCHEMBL10617106 0.82 KMT2A (0.51) LMNAOPRM1OPRL1OGFRL1KMT2A
SCHEMBL6245939 0.80 MAPKAPK2 (0.54) LMNAKDM4EMAPKAPK2TSHRALDH1A1
SCHEMBL12592476 0.79 LMNA (0.60) LMNAOPRM1OPRL1OGFRL1KMT2A
Hydrochloric Acid SCHEMBL6354640 0.79 MAPKAPK2 (0.53) LMNAKMT2AKDM4EMAPKAPK2TSHR
SCHEMBL10484393 0.79 KMT2A (0.50) LMNAOPRM1OPRL1OGFRL1KMT2A
SCHEMBL274568 0.77 OPRM1 (0.60) LMNAOPRM1OPRL1OGFRL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111303148-B 1-substituted beta-carboline derivatives and application thereof 南京农业大学 2022-08-30 CN disclosed
CN-111303148-A 1-substituted β -carboline derivatives and application thereof 南京农业大学 2020-06-19 CN disclosed
US-5256533-A Preincubating sample with an alpha-2-inhibitor; comparing fluorescence in test to control tissues BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 1993-10-26 US disclosed
WO-1991014184-A1 BETA CARBOLINES AS VITAL STAINS FOR NEUROTRANSMITTER SYSTEMS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1991-09-19 WO disclosed