SCHEMBL9484205

SCHEMBL9484205

CC1CC(C)(C)c2cc(C#Cc3ccc(C(=O)O)cc3)ccc2C1(C)C

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RARB P10826 20/20 0.67
RARG P13631 20/20 0.67
RARA P10276 18/20 0.67
CYP26A1 O43174 1/20 0.67
CYP3A4 P08684 1/20 0.67
CRABP2 P29373 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776432 0.82 RARB (0.63) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9483506 0.82 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8776480 0.81 RARB (0.83) RARBRARGRARACYP26A1CYP3A4
SCHEMBL3302926 0.81 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL29353973 0.81 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9329536 0.78 RARB (0.57) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8437077 0.77 RARB (0.66) RARBRARGRARACYP26A1CYP3A4
SCHEMBL12620671 0.76 RXRA (0.42) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8866611 0.75 RARB (0.63) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8631781 0.75 RARB (0.63) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256694-A For skin disorders; carcinomas BASF AKTIENGESELLSCHAFT (DE) 1993-10-26 US disclosed
US-5126371-A Precancerous skin conditions, acne, psoriasis BASF AKTEINGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-4994489-A Ester derivatives of diarylacetylenes, their compositions and their use in acne treatment BASF AKTIENGESELLSCHAFT 1991-02-19 US disclosed
US-4806558-A Diarylacetylenes and their use in treating acne BASF AKTIENGESELLSCHAFT (DE) 1989-02-21 US disclosed