SCHEMBL9484455

SCHEMBL9484455

CC1(C)CCC(C)(C)c2cc(C#Cc3ccc(C(N)=O)cc3)ccc21

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARB P10826 12/20 0.76
RARG P13631 12/20 0.76
RARA P10276 7/20 0.76
CYP26A1 O43174 3/20 0.76
CYP3A4 P08684 2/20 0.76
CRABP2 P29373 1/20 0.76
RXRA P19793 10/20 0.49
RXRB P28702 9/20 0.49
RXRG P48443 6/20 0.49
CYP26B1 Q9NR63 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19697334 0.87 RARB (0.78) RARBRARGRARACYP26A1CYP3A4
SCHEMBL3302926 0.87 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL29353973 0.87 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7752077 0.84 RARB (0.55) RARBRARGRARACYP26A1CYP3A4
SCHEMBL2195010 0.82 RXRA (0.63) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9484975 0.80 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9484589 0.78 RARB (0.65) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8776480 0.78 RARB (0.83) RARBRARGRARACYP26A1CYP3A4
SCHEMBL31046815 0.77 RARB (0.77) RARBRARGRARACYP26A1CYP3A4
SCHEMBL20587536 0.77 RARB (0.77) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256694-A For skin disorders; carcinomas BASF AKTIENGESELLSCHAFT (DE) 1993-10-26 US disclosed
US-5126371-A Precancerous skin conditions, acne, psoriasis BASF AKTEINGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-4994489-A Ester derivatives of diarylacetylenes, their compositions and their use in acne treatment BASF AKTIENGESELLSCHAFT 1991-02-19 US disclosed
EP-0176034-B1 DIARYL ACETYLENES, THEIR PREPARATION AND USE BASF Aktiengesellschaft (DE) 1989-08-30 EP disclosed
US-4806558-A Diarylacetylenes and their use in treating acne BASF AKTIENGESELLSCHAFT (DE) 1989-02-21 US disclosed
EP-0176034-A2 Diaryl acetylenes, their preparation and use BASF Aktiengesellschaft (DE) 1986-04-02 EP disclosed