SCHEMBL9485648

SCHEMBL9485648

Cc1nc(N)nc(N)c1-c1ccc(Cl)c([N+](=O)[O-])c1

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NCOA1 Q15788 1/20 0.72
NCOA3 Q9Y6Q9 1/20 0.72
DHFR P00374 1/20 0.60
CYP2D6 P10635 2/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HIF1A Q16665 1/20 0.53
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6359292 0.84 NCOA1 (1.00) NCOA1NCOA3CYP2D6
SCHEMBL6049524 0.80 NCOA1 (0.50) NCOA1NCOA3DHFRCYP2D6TP53
Metoprine SCHEMBL3681 0.80 NPC1 (0.54) NCOA1NCOA3DHFRCYP2D6TP53
Metoprine SCHEMBL29463675 0.80 NPC1 (0.54) NCOA1NCOA3DHFRCYP2D6TP53
Metoprine SCHEMBL4529657 0.79 NPC1 (0.53) NCOA1NCOA3DHFRCYP2D6TP53
SCHEMBL9566530 0.77 DHFR (0.60) NCOA1NCOA3DHFRMEN1ALDH1A1
SCHEMBL27612645 0.76 DHFR (0.60) NCOA1NCOA3DHFRCYP2D6TP53
SCHEMBL6049511 0.76 NCOA1 (0.46) NCOA1NCOA3DHFRCYP2D6TP53
SCHEMBL10999078 0.76 ALDH1A1 (0.48) NCOA1NCOA3DHFRCYP2D6TP53
SCHEMBL6049617 0.76 NCOA1 (0.45) NCOA1NCOA3DHFRCYP2D6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290558-B1 ANTIFOLATE AGENTS BTG INTERNATIONAL LIMITED (GB) 1993-06-16 EP disclosed
US-4992444-A Antitumor agents, skin disorders BRITISH TECHNOLOGY GROUP LIMITED (GB) 1991-02-12 US disclosed
EP-0290558-A1 ANTIFOLATE AGENTS. STEVENS MALCOLM FRANCIS GRAHAM (GB) 1988-11-17 EP disclosed
WO-1988004293-A1 ANTIFOLATE AGENTS STEVENS MALCOLM FRANCIS GRAHAM (GB) 1988-06-16 WO disclosed
EP-0147443-A1 PYRIMIDINE DERIVATIVES Aston Molecules Limited (GB) 1985-07-10 EP disclosed
WO-1984004746-A1 PYRIMIDINE DERIVATIVES UNIV BIRMINGHAM (GB) 1984-12-06 WO disclosed