SCHEMBL948567

SCHEMBL948567

CC(C)(C)OC(=O)CC1c2cc3cc(/C(N)=N\O)ccc3n2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.32
NR1H3 Q13133 2/20 0.32
CHEK2 O96017 4/20 0.32
GPR119 Q8TDV5 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
SETD7 Q8WTS6 1/20 0.31
HDAC4 P56524 1/20 0.31
NOD2 Q9HC29 1/20 0.31
NOD1 Q9Y239 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL948569 1.00 NR1H2 (0.32) NR1H2NR1H3CHEK2GPR119MEN1
SCHEMBL948843 0.84 ESR2 (0.38) NR1H2NR1H3GPR119MEN1KMT2A
SCHEMBL948658 0.83 S1PR1 (0.40)
SCHEMBL948657 0.83 S1PR1 (0.40)
SCHEMBL949210 0.81 S1PR1 (0.41)
SCHEMBL949211 0.81 S1PR1 (0.41)
SCHEMBL949792 0.76 S1PR1 (0.34)
SCHEMBL3746518 0.73 S1PR1 (0.40)
SCHEMBL3401067 0.73 S1PR1 (0.40)
SCHEMBL948764 0.69 S1PR1 (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed