SCHEMBL9490489

SCHEMBL9490489

CNC(=S)[C@]1(c2cccnc2)CCCC[C@H]1OC(=O)COc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
GAA P10253 2/20 0.43
NOTUM Q6P988 1/20 0.39
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CPT1A P50416 4/20 0.37
CPT1B Q92523 3/20 0.37
CPT2 P23786 3/20 0.37
ITGA4 P13612 2/20 0.36
ITGB7 P26010 2/20 0.36
P2RX7 Q99572 1/20 0.36
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CNR2 P34972 1/20 0.34
VNN1 O95497 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9490262 0.89 ITGA4 (0.36) KDM4EGAAALDH1A1ITGA4ITGB7
SCHEMBL9490652 0.87 MEN1 (0.40) ALDH1A1ITGA4ITGB7P2RX7
SCHEMBL9491683 0.87 P2RX7 (0.35) KDM4EGAAALDH1A1ITGA4ITGB7
SCHEMBL10432053 0.87 MEN1 (0.40) ALDH1A1ITGA4ITGB7P2RX7
SCHEMBL10431870 0.87 P2RX7 (0.35) KDM4EGAAALDH1A1ITGA4ITGB7
SCHEMBL9491888 0.87 ITGA4 (0.37) GAAALDH1A1ITGA4ITGB7P2RX7
SCHEMBL9491885 0.86 CYP1A2 (0.39) KDM4EMAPTALDH1A1ITGA4ITGB7
SCHEMBL9521814 0.86 CYP1A2 (0.39) KDM4EMAPTALDH1A1ITGA4ITGB7
SCHEMBL9520740 0.85 ITGA4 (0.36) GAAALDH1A1ITGA4ITGB7P2RX7
SCHEMBL9491001 0.85 GAA (0.37) GAAALDH1A1ITGA4ITGB7P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5246950-A Smooth muscle disorders RHONE-POULENC SANTE (FR) 1993-09-21 US disclosed
EP-0390693-B1 THIOFORMAMIDE DERIVATIVES RHONE-POULENC SANTE (FR) 1993-08-25 EP disclosed
EP-0390693-A1 Thioformamide derivatives RHONE-POULENC SANTE (FR) 1990-10-03 EP disclosed