SCHEMBL9490860

SCHEMBL9490860

COc1ccc(C(C=O)n2ccnc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.66
CYP26A1 O43174 2/20 0.50
KMT2A Q03164 2/20 0.48
CYP17A1 P05093 2/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
P4HB P07237 1/20 0.46
CYP24A1 Q07973 2/20 0.45
MEN1 O00255 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5721926 0.83 CYP17A1 (0.51) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1
SCHEMBL11242107 0.80 CYP19A1 (0.63) CYP19A1CYP26A1KMT2ACYP17A1CYP24A1
SCHEMBL7387804 0.80 CYP19A1 (0.61) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1
SCHEMBL27618666 0.80 CYP19A1 (0.76) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1
SCHEMBL19054896 0.78 CYP19A1 (0.73) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1
SCHEMBL11287252 0.78 CYP17A1 (0.74) CYP19A1KMT2ACYP17A1CYP11B1CYP11B2
SCHEMBL11245762 0.77 CYP19A1 (0.66) CYP19A1CYP17A1CYP11B1CYP11B2
SCHEMBL19999188 0.76 CYP19A1 (0.69) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1
SCHEMBL11436593 0.75 CYP26A1 (0.52) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1
SCHEMBL19999180 0.75 CYP19A1 (0.88) CYP19A1CYP26A1KMT2ACYP17A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5236944-A C1-4 alkyl(4-(2-(4-C1-4-alkylphenyl)-2(1H-imidazol-1-ylmethyl) -1,3-dioxolan-4-ylemthlthio)phenyl)carbamate JANSSEN PHARMACEUTICA N.V. (BE) 1993-08-17 US disclosed
EP-0335446-A2 Agents for treating neoplasms JANSSEN PHARMACEUTICA N.V. (BE) 1989-10-04 EP disclosed