SCHEMBL9493360

SCHEMBL9493360

COc1ccc(C2CN3CCC2CC3)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.61
KDM1A O60341 2/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
HTR3A P46098 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
DRD2 P14416 1/20 0.43
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9495813 0.91 CHRNA7 (0.55) CHRNA7MEN1KMT2ACHRM2CHRM4
SCHEMBL9494114 0.83 CHRNA7 (0.51) CHRNA7HTR3ACHRM2CHRM4CHRM5
SCHEMBL9496249 0.81 CHRNA7 (0.58) CHRNA7HTR3ADRD2HTR2C
SCHEMBL9492454 0.79 CHRNA7 (0.51) CHRNA7
SCHEMBL11300641 0.77 CHRNA7 (0.67) CHRNA7KDM1ACHRM2CHRM4CHRM5
SCHEMBL9431069 0.77 CHRNA7 (0.67) CHRNA7CHRM2CHRM4CHRM5CHRM1
SCHEMBL9492423 0.76 MTNR1A (0.46) CHRNA7HTR3A
SCHEMBL9494509 0.76 MEN1 (0.47) CHRNA7HTR3AMEN1KMT2A
SCHEMBL9431093 0.76 CHRNB2 (0.46) CHRNA7
SCHEMBL9431625 0.76 CHRNA7 (0.49) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0412797-A2 The therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes MERCK SHARP & DOHME LTD. (GB) 1991-02-13 EP claimed
US-5177084-A 1-Azabicycles, Treating Mental Disorders MERCK SHARP & DOHME LTD. (GB) 1993-01-05 US disclosed
EP-0492904-A1 Substituted benzene derivatives for use in the treatment of glaucoma MERCK SHARP & DOHME LTD. (GB) 1992-07-01 EP disclosed
EP-0412797-A2 The therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes MERCK SHARP & DOHME LTD. (GB) 1991-02-13 EP disclosed
US-4292190-A ANTIFREEZES FOR COOLING SYSTEMS OF INTERNAL COMBUSTION ENGINES BASF WYANDOTTE CORPORATION (US) 1981-09-29 US disclosed