SCHEMBL9496249

SCHEMBL9496249

COc1cccc(C2CN3CCC2CC3)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.58
CHRNB2 P17787 1/20 0.51
CHRNA4 P43681 1/20 0.51
HTR3A P46098 1/20 0.51
HTR2C P28335 4/20 0.49
HTR2A P28223 2/20 0.49
HTR2B P41595 2/20 0.49
DPP4 P27487 1/20 0.48
DRD2 P14416 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9494451 0.93 CHRNA7 (0.49) CHRNA7CHRNB2CHRNA4HTR3AHTR2C
Oxalic Acid SCHEMBL9494045 0.92 CHRNA7 (0.54) CHRNA7CHRNB2CHRNA4HTR3AHTR2C
SCHEMBL9493175 0.84 DRD2 (0.51) HTR2CHTR2AHTR2BDPP4DRD2
SCHEMBL9494114 0.84 CHRNA7 (0.51) CHRNA7CHRNB2CHRNA4HTR3A
Cadaverine Tartrate SCHEMBL9493533 0.81 GRIN2B (0.42) CHRNA7CHRNB2CHRNA4HTR3ADPP4
SCHEMBL9493360 0.81 CHRNA7 (0.61) CHRNA7HTR3AHTR2CDRD2
Oxalic Acid SCHEMBL9494495 0.79 DRD2 (0.46) DRD2
SCHEMBL9431093 0.78 CHRNB2 (0.46) CHRNA7CHRNB2CHRNA4
SCHEMBL9494509 0.78 MEN1 (0.47) CHRNA7CHRNB2CHRNA4HTR3A
SCHEMBL9492454 0.77 CHRNA7 (0.51) CHRNA7DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0412797-A2 The therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes MERCK SHARP & DOHME LTD. (GB) 1991-02-13 EP claimed
US-5177084-A 1-Azabicycles, Treating Mental Disorders MERCK SHARP & DOHME LTD. (GB) 1993-01-05 US disclosed
EP-0412797-A2 The therapeutic use of substituted benzenes, formulations thereof and novel substituted benzenes MERCK SHARP & DOHME LTD. (GB) 1991-02-13 EP disclosed