SCHEMBL9494868

SCHEMBL9494868

O=C1c2c(Cl)cccc2OCN1CCO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
ACKR3 P25106 2/20 0.32
ITGB1 P05556 4/20 0.32
ITGA2 P17301 4/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
TSHR P16473 1/20 0.32
HEXA P06865 1/20 0.32
HEXB P07686 1/20 0.32
WEE1 P30291 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
CHEK1 O14757 1/20 0.32
HSD17B10 Q99714 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9491320 0.87 TSHR (0.33) DRD2ACKR3ITGB1ITGA2TSHR
SCHEMBL8980622 0.83 PARP1 (0.43) PARP1PARP2SIRT2SIRT1HEXA
SCHEMBL9493171 0.81 ALDH1A1 (0.36) PARP1ACKR3TSHR
SCHEMBL9492003 0.78 PTK2 (0.30)
SCHEMBL6947117 0.76 TSHR (0.41) PARP1PARP2SIRT1TSHRHEXA
SCHEMBL8573189 0.71 MAOB (0.40) MAPTNPSR1
SCHEMBL8980735 0.71 DPP4 (0.39) NPSR1
SCHEMBL8368757 0.70 KDM4E (0.35) PARP1PARP2TSHRHEXAHEXB
SCHEMBL8980753 0.69 DPP4 (0.36)
SCHEMBL8578943 0.68 PRMT5 (0.39) SIRT1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5189034-A Vasodilating, antianginal agents ITALFARMACO S.P.A. (IT) 1993-02-23 US disclosed
EP-0490183-A1 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity ITALFARMACO S.p.A. (IT) 1992-06-17 EP disclosed