SCHEMBL949658

SCHEMBL949658

Fc1c(F)c(F)c(-c2c(F)c(F)c(F)c(F)c2C#Cc2ccccc2)c(F)c1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.50
MAPT P10636 2/20 0.40
GRM5 P41594 6/20 0.38
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
NPC1 O15118 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HSD17B10 Q99714 1/20 0.36
KCNH2 Q12809 1/20 0.35
THPO P40225 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6519831 0.94 APP (0.52) APPMAPTGRM5CYP1A2CYP3A4
SCHEMBL952971 0.87 APP (0.60) APPMAPTGRM5CYP1A2CYP3A4
SCHEMBL10300049 0.84 APP (0.63) APPMAPTGRM5CYP1A2CYP3A4
SCHEMBL17711134 0.75 APP (0.50) APPMAPTGRM5CYP1A2CYP3A4
SCHEMBL10300067 0.74 APP (0.41) APPMAPTGRM5CYP2C19KDM4E
SCHEMBL10300107 0.74 APP (0.41) APPMAPTGRM5CYP2C19KDM4E
SCHEMBL3796509 0.74 APP (0.80) APPMAPTGRM5CYP1A2CYP3A4
SCHEMBL5134940 0.71 APP (0.57) APPMAPTGRM5CYP1A2CYP3A4
Diphenylacetylene SCHEMBL960609 0.71 APP (1.00) APPMAPTGRM5CYP1A2CYP3A4
Diphenylacetylene SCHEMBL29188592 0.71 APP (1.00) APPMAPTGRM5CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519080-B2 Crosslinkable prepolymer, its production process and its uses ASAHI GLASS COMPANY, LIMITED (JP) 2013-08-27 US claimed
US-9575246-B2 Prepolymer, curable material, coating composition, non-linear optical material, optical waveguide and light control device ASAHI GLASS COMPANY, LIMITED (JP) 2017-02-21 US disclosed
EP-2792665-B1 LIQUID REPELLENT COMPOSITION, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT ASAHI GLASS CO LTD (JP) 2016-08-03 EP disclosed
EP-2266792-B1 ELECTRET AND ELECTROSTATIC INDUCTION CONVERSION DEVICE ASAHI GLASS CO LTD (JP) 2016-05-04 EP disclosed
EP-2889684-A1 PREPOLYMER, CURABLE MATERIAL, COATING COMPOSITION, NON-LINEAR OPTICAL MATERIAL, OPTICAL WAVEGUIDE AND LIGHT CONTROL DEVICE Asahi Glass Company, Limited (JP) 2015-07-01 EP disclosed
US-20150153509-A1 PREPOLYMER, CURABLE MATERIAL, COATING COMPOSITION, NON-LINEAR OPTICAL MATERIAL, OPTICAL WAVEGUIDE AND LIGHT CONTROL DEVICE ASAHI GLASS COMPANY, LIMITED (JP) 2015-06-04 US disclosed
EP-2810962-A1 COMPOUND, POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LYOPHILIC REGIONS AND LYOPHOBIC REGIONS, AND METHOD FOR PRODUCING SAME Asahi Glass Company, Limited (JP) 2014-12-10 EP disclosed
EP-2792665-A1 LIQUID REPELLENT COMPOUND, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN WITH LYOPHILIC REGION AND LIQUID REPELLENT REGION, AND METHOD FOR PRODUCING SAME Asahi Glass Company, Limited (JP) 2014-10-22 EP disclosed
US-20140295149-A1 LIQUID REPELLENT COMPOSITION, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT ASAHI GLASS COMPANY, LIMITED (JP) 2014-10-02 US disclosed
US-20140287200-A1 COMPOUND, POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT ASAHI GLASS COMPANY, LIMITED (JP) 2014-09-25 US disclosed
US-20100144914-A1 CROSSLINKABLE FLUORINATED AROMATIC PREPOLYMER AND ITS USES ASAHI GLASS COMPANY, LIMITED (JP) 2010-06-10 US disclosed
EP-1669389-B1 CROSSLINKABLE FLUOROAROMATIC PREPOLYMER AND USE THEREOF ASAHI GLASS CO LTD (JP) 2009-08-26 EP disclosed
US-20090081376-A1 CROSSLINKABLE PREPOLYMER, ITS PRODUCTION PROCESS AND ITS USES ASAHI GLASS COMPANY, LIMITED (JP) 2009-03-26 US disclosed
EP-2025698-A1 CROSSLINKABLE PREPOLYMER, PROCESS FOR PRODUCTION THEREOF, AND USE THEREOF Asahi Glass Company, Limited (JP) 2009-02-18 EP disclosed
US-20090017265-A1 NEGATIVE PHOTOSENSITIVE FLUORINATED AROMATIC RESIN COMPOSITION ASAHI GLASS COMPANY LIMITED (JP) 2009-01-15 US disclosed
EP-1995635-A1 NEGATIVE-TYPE PHOTOSENSITIVE FLUORINATED AROMATIC RESIN COMPOSITION Asahi Glass Company, Limited (JP) 2008-11-26 EP disclosed
US-20060173129-A1 Crosslinkable fluorinated aromatic prepolymer and its uses ASAHI GLASS COMPANY, LIMITED (JP) 2006-08-03 US disclosed
EP-1669389-A1 CROSSLINKABLE FLUOROAROMATIC PREPOLYMER AND USE THEREOF ASAHI GLASS COMPANY LTD. (JP) 2006-06-14 EP disclosed
US-6881811-B2 Improved heat resistance and low relative permittivity; insulating films for electronic devices/multilayerd wiring boards ASAHI GLASS COMPANY, LIMITED (JP) 2005-04-19 US disclosed
US-20040147710-A1 Improved heat resistance and low relative permittivity; insulating films for electronic devices/multilayerd wiring boards ASAHI GLASS COMPANY LIMITED (JP) 2004-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140295149-A1 LIQUID REPELLENT COMPOSITION, LIQUID REPELLENT POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT CHRM1, C5, SETDB1 APP 1777/4885MAPT 701/4885GRM5 1012/4885
US-20140287200-A1 COMPOUND, POLYMER, CURABLE COMPOSITION, COATING COMPOSITION, ARTICLE HAVING CURED FILM, ARTICLE HAVING PATTERN OF LIQUID-PHILIC REGION AND LIQUID REPELLENT REGION, AND PROCESS FOR PRODUCING IT H1-0, DNMT1, BMI1 APP 1763/4885MAPT 954/4885GRM5 1794/4885
US-20100144914-A1 CROSSLINKABLE FLUORINATED AROMATIC PREPOLYMER AND ITS USES AFF1, AFF2, FPR1 APP 2563/4885MAPT 3309/4885GRM5 4580/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.