SCHEMBL9497323

SCHEMBL9497323

Clc1ccc(C(Cl)(Cl)Cl)c2nc(C(Cl)(Cl)Cl)cc(Cl)c12

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.38
CYP3A4 P08684 2/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
FABP4 P15090 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9493285 0.90 FABP4 (0.37) TSHRCYP3A4MAPK1TDP1ALDH1A1
SCHEMBL11100320 0.87 TSHR (0.41) TSHRCYP3A4ALDH1A1LMNAFABP4
SCHEMBL9493505 0.81 CYP3A4 (0.36) TSHRCYP3A4ALDH1A1NPSR1
SCHEMBL10508928 0.79 NT5E (0.39) ALDH1A1LMNAFABP4NPSR1
SCHEMBL9492503 0.77 CYP3A4 (0.40) TSHRCYP3A4MAPK1TDP1ALDH1A1
SCHEMBL21144535 0.71 MAPT (0.39) TSHRCYP3A4TDP1ALDH1A1LMNA
SCHEMBL9493152 0.70 NR4A2 (0.46) TSHRCYP3A4TDP1ALDH1A1LMNA
SCHEMBL11099839 0.69 MAPT (0.35) TSHRCYP3A4TDP1LMNA
SCHEMBL9493489 0.68 ALDH1A1 (0.43) TSHRCYP3A4ALDH1A1LMNANPSR1
SCHEMBL10506369 0.68 CYP3A4 (0.38) TSHRCYP3A4ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0113432-B1 CHLOROMETHYL QUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE ALKALOIDA VEGYéSZETI GYáR (HU) 1993-03-17 EP claimed