SCHEMBL9497776

SCHEMBL9497776

COc1ccc(C#Cc2ccc(C)cn2)c(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.41
AAK1 Q2M2I8 2/20 0.35
SYK P43405 1/20 0.34
AURKB Q96GD4 1/20 0.34
INCENP Q9NQS7 1/20 0.34
ACHE P22303 1/20 0.33
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
SLC22A12 Q96S37 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10511880 0.90 GRM5 (0.38) GRM5AAK1SYKAURKBINCENP
SCHEMBL9497092 0.87 GRM5 (0.38) GRM5SLC22A12
SCHEMBL9498411 0.84 GRM5 (0.36) GRM5MEN1GAAMAPTKMT2A
SCHEMBL9496170 0.83 GRM5 (0.35) GRM5GAAMAPTRAB9A
SCHEMBL9500393 0.82 ACACB (0.35) GRM5AAK1
SCHEMBL9497011 0.82 ALDH1A1 (0.35) GRM5GAAMAPT
SCHEMBL9496861 0.80 ACACB (0.38) GRM5MEN1MAPTRAB9AKMT2A
SCHEMBL9495259 0.78 CASP3 (0.41) MEN1MAPTRAB9AKMT2A
SCHEMBL4147152 0.78 GRM5 (0.55) GRM5MEN1RAB9AKMT2A
SCHEMBL9496334 0.77 CASP3 (0.45) MEN1GAAMAPTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed