SCHEMBL949880

SCHEMBL949880

Cc1c(C)n(-c2ccc(C#N)c(Br)c2)c2cccc(-c3cnc4ccccc4c3)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.36
HSP90AA1 P07900 5/20 0.36
ABCG2 Q9UNQ0 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP11 Q9NR21 1/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
PIK3CA P42336 4/20 0.34
MTOR P42345 3/20 0.34
PIK3C2A O00443 2/20 0.34
PIK3C2B O00750 2/20 0.34
PIK3CD O00329 2/20 0.34
CHEK1 O14757 1/20 0.34
ABCB11 O95342 1/20 0.34
CSF1R P07333 1/20 0.34
MET P08581 1/20 0.34
PIK3R1 P27986 1/20 0.34
LTK P29376 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2183119 0.87 BIRC5 (0.37) BIRC5HSP90AA1ABCG2PIK3CAMTOR
SCHEMBL951332 0.84 BIRC5 (0.37) BIRC5HSP90AA1ABCG2PARP10PARP11
SCHEMBL425541 0.83 HSP90AA1 (0.51) BIRC5HSP90AA1ABCG2ALDH1A1NPC1
SCHEMBL952602 0.83 HSP90AA1 (0.51) BIRC5HSP90AA1ABCG2ALDH1A1NPC1
SCHEMBL2183124 0.82 BIRC5 (0.38) BIRC5HSP90AA1ABCG2PIK3CAMTOR
SCHEMBL949653 0.80 HSP90AA1 (0.56) HSP90AA1
SCHEMBL420055 0.78 HSP90AA1 (0.49) BIRC5HSP90AA1ABCG2ALDH1A1NPC1
SCHEMBL950675 0.78 HSP90AA1 (0.49) BIRC5HSP90AA1ABCG2ALDH1A1NPC1
SCHEMBL1394564 0.78 HSP90AA1 (0.46) BIRC5HSP90AA1NPC1MAPTRAB9A
SCHEMBL2181737 0.76 CYP11B1 (0.42) HSP90AA1NPC1MAPTRAB9APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011004132-A1 NOVEL HSP90-INHIBITING INDOLE DERIVATIVES, COMPOSITIONS CONTAINING SAID DERIVATIVES, AND USE THEREOF SANOFI-AVENTIS (FR) 2011-01-13 WO disclosed