SCHEMBL950675

SCHEMBL950675

N#Cc1ccc(-n2ccc3c(-c4cnc5ccccc5c4)cccc32)cc1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.49
BIRC5 O15392 1/20 0.38
PDGFRB P09619 2/20 0.35
PDGFRA P16234 2/20 0.35
CYP19A1 P11511 1/20 0.35
PIK3CA P42336 3/20 0.35
MTOR P42345 3/20 0.35
PIK3C2A O00443 2/20 0.35
PIK3C2B O00750 2/20 0.35
PIK3CD O00329 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 2/20 0.35
PRKDC P78527 2/20 0.35
ATM Q13315 2/20 0.35
MET P08581 2/20 0.35
CHEK1 O14757 1/20 0.35
ABCB11 O95342 1/20 0.35
CSF1R P07333 1/20 0.35
PIK3R1 P27986 1/20 0.35
LTK P29376 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693085 0.85 HSP90AA1 (0.36) HSP90AA1BIRC5PDGFRBPDGFRA
SCHEMBL950332 0.85 HSP90AA1 (0.51) HSP90AA1BIRC5PDGFRBPDGFRACYP19A1
SCHEMBL420055 0.84 HSP90AA1 (0.49) HSP90AA1BIRC5PDGFRBPDGFRAPIK3CA
SCHEMBL951332 0.83 BIRC5 (0.37) HSP90AA1BIRC5PDGFRBPDGFRAPIK3CA
SCHEMBL2183124 0.82 BIRC5 (0.38) HSP90AA1BIRC5PDGFRBPDGFRAPIK3CA
SCHEMBL952602 0.82 HSP90AA1 (0.51) HSP90AA1BIRC5PIK3CAMTORPIK3C2A
SCHEMBL2183119 0.82 BIRC5 (0.37) HSP90AA1BIRC5PDGFRBPDGFRAPIK3CA
SCHEMBL422414 0.81 BIRC5 (0.41) BIRC5PDGFRBPDGFRAPIK3CAMTOR
SCHEMBL951938 0.79 HSP90AA1 (0.74) HSP90AA1
SCHEMBL949880 0.78 BIRC5 (0.36) HSP90AA1BIRC5PDGFRBPDGFRAPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011004132-A1 NOVEL HSP90-INHIBITING INDOLE DERIVATIVES, COMPOSITIONS CONTAINING SAID DERIVATIVES, AND USE THEREOF SANOFI-AVENTIS (FR) 2011-01-13 WO disclosed