SCHEMBL951332

SCHEMBL951332

Cc1cc2c(-c3cnc4ccccc4c3)cccc2n1-c1ccc(C#N)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.37
PIK3CA P42336 5/20 0.36
MTOR P42345 4/20 0.36
PIK3CD O00329 3/20 0.36
PIK3C2A O00443 2/20 0.36
PIK3C2B O00750 2/20 0.36
MET P08581 2/20 0.36
PIK3CB P42338 2/20 0.36
PIK3CG P48736 2/20 0.36
PRKDC P78527 2/20 0.36
ATM Q13315 2/20 0.36
CHEK1 O14757 1/20 0.36
ABCB11 O95342 1/20 0.36
CSF1R P07333 1/20 0.36
PIK3R1 P27986 1/20 0.36
LTK P29376 1/20 0.36
CDK7 P50613 1/20 0.36
NEK2 P51955 1/20 0.36
JAK3 P52333 1/20 0.36
LIMK1 P53667 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2183124 0.87 BIRC5 (0.38) BIRC5PIK3CAMTORPIK3CDPIK3C2A
SCHEMBL2183119 0.86 BIRC5 (0.37) BIRC5PIK3CAMTORPIK3CDPIK3C2A
SCHEMBL947823 0.85 PIK3CA (0.40) PIK3CAMTORPIK3CDPIK3C2APIK3C2B
SCHEMBL949880 0.84 BIRC5 (0.36) BIRC5PIK3CAMTORPIK3CDPIK3C2A
SCHEMBL420055 0.83 HSP90AA1 (0.49) BIRC5PIK3CAMTORPIK3CDPIK3C2A
SCHEMBL950675 0.83 HSP90AA1 (0.49) BIRC5PIK3CAMTORPIK3CDPIK3C2A
SCHEMBL425541 0.80 HSP90AA1 (0.51) BIRC5ABCG2ALDH1A1NPC1MAPT
SCHEMBL952602 0.80 HSP90AA1 (0.51) BIRC5PIK3CAMTORPIK3CDPIK3C2A
SCHEMBL954168 0.80 HSP90AA1 (0.55) HSP90AA1
SCHEMBL422414 0.80 BIRC5 (0.41) BIRC5PIK3CAMTORPIK3CDPIK3C2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011004132-A1 NOVEL HSP90-INHIBITING INDOLE DERIVATIVES, COMPOSITIONS CONTAINING SAID DERIVATIVES, AND USE THEREOF SANOFI-AVENTIS (FR) 2011-01-13 WO disclosed