SCHEMBL9499272

SCHEMBL9499272

Cc1cc(NCc2ccc(-c3ccccc3-c3nnn(C(c4ccccc4)(c4ccccc4)c4ccccc4)n3)cc2)c(Cl)c(C)n1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 9/20 0.62
AGTR2 P50052 8/20 0.62
USP1 O94782 1/20 0.36
WDR48 Q8TAF3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9496626 0.90 AGTR1 (0.62) AGTR1AGTR2USP1WDR48
SCHEMBL9494062 0.86 AGTR1 (0.66) AGTR1AGTR2
SCHEMBL9494452 0.83 AGTR1 (0.65) AGTR1AGTR2
SCHEMBL9495030 0.81 AGTR1 (0.47) AGTR1AGTR2
SCHEMBL9499263 0.79 AGTR1 (0.37) AGTR1AGTR2
SCHEMBL9494926 0.78 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL9494775 0.77 AGTR1 (0.65) AGTR1AGTR2
SCHEMBL9495741 0.77 AGTR1 (0.65) AGTR1AGTR2
SCHEMBL9454713 0.77 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL9454802 0.76 AGTR1 (0.42) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5236937-A Treating hypertension, congestive heart failure IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-08-17 US disclosed
EP-0499415-A1 Pyridine and quinoline derivatives, processes for their manufacture and their use as angiotensin II antagonists ZENECA LIMITED (GB) 1992-08-19 EP disclosed